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Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50013309
TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128951(4-Ethyl-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50: <3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128955(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-isobutoxy...)
Affinity DataIC50: <3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128960(CHEMBL59817 | N-{(S)-1-[2-(4-Benzyloxy-phenylamino...)
Affinity DataIC50: <3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128957(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-cyclopent...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128964(CHEMBL58179 | N-{(S)-1-[2-(4-Isobutoxy-phenylamino...)
Affinity DataIC50: <3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128962(CHEMBL294260 | N-{(S)-1-[2-(4-Cyclopentylmethoxy-p...)
Affinity DataIC50: <3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128965(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-cyclohexy...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113674(4-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128950(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-methoxy-p...)
Affinity DataIC50: <30nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128949(CHEMBL292472 | N-{(S)-1-[2-(4-Methoxy-phenylamino)...)
Affinity DataIC50: <30nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128951(4-Ethyl-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM19545((2S)-N-{2-[(4-methoxyphenyl)amino]ethyl}-4-methyl-...)
Affinity DataIC50: <32nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128953(CHEMBL64178 | {(S)-1-[2-(4-Isobutoxy-phenylamino)-...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128971(CHEMBL304669 | {(S)-1-[2-(4-Cyclohexyloxy-phenylam...)
Affinity DataIC50:  43nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128949(CHEMBL292472 | N-{(S)-1-[2-(4-Methoxy-phenylamino)...)
Affinity DataIC50:  44nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128954(CHEMBL291587 | {(S)-1-[2-(4-Cyclopentylmethoxy-phe...)
Affinity DataIC50:  49nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128961(CHEMBL300379 | {(S)-1-[2-(4-Benzyloxy-phenylamino)...)
Affinity DataIC50:  54nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128952(CHEMBL64367 | {(S)-1-[2-(4-Cyclopropylmethoxy-phen...)
Affinity DataIC50:  69nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM19545((2S)-N-{2-[(4-methoxyphenyl)amino]ethyl}-4-methyl-...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128959(CHEMBL303517 | {(S)-1-[2-(4-Cyclopentyloxy-phenyla...)
Affinity DataIC50:  81nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128950(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-methoxy-p...)
Affinity DataIC50:  90nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128969(3-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128967(CHEMBL64546 | N-{(S)-1-[2-(4-Methoxy-phenylamino)-...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128968(((S)-3-Methyl-1-{2-[4-(pyridin-4-ylmethoxy)-phenyl...)
Affinity DataIC50:  152nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128950(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-methoxy-p...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128956(((S)-3-Methyl-1-{2-[4-(tetrahydro-pyran-4-yloxy)-p...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128970(CHEMBL62207 | {(S)-3-Methyl-1-[2-(4-phenoxy-phenyl...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128967(CHEMBL64546 | N-{(S)-1-[2-(4-Methoxy-phenylamino)-...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM19545((2S)-N-{2-[(4-methoxyphenyl)amino]ethyl}-4-methyl-...)
Affinity DataIC50:  372nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128969(3-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  419nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128969(3-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  470nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128962(CHEMBL294260 | N-{(S)-1-[2-(4-Cyclopentylmethoxy-p...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128964(CHEMBL58179 | N-{(S)-1-[2-(4-Isobutoxy-phenylamino...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128967(CHEMBL64546 | N-{(S)-1-[2-(4-Methoxy-phenylamino)-...)
Affinity DataIC50:  490nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128962(CHEMBL294260 | N-{(S)-1-[2-(4-Cyclopentylmethoxy-p...)
Affinity DataIC50:  580nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128949(CHEMBL292472 | N-{(S)-1-[2-(4-Methoxy-phenylamino)...)
Affinity DataIC50:  580nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128964(CHEMBL58179 | N-{(S)-1-[2-(4-Isobutoxy-phenylamino...)
Affinity DataIC50:  580nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128951(4-Ethyl-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  660nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113674(4-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128972(((S)-1-{2-[4-(2-Imidazol-1-yl-ethoxy)-phenylamino]...)
Affinity DataIC50:  855nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128966(((S)-3-Methyl-1-{2-[4-(2-pyrrolidin-1-yl-ethoxy)-p...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128963(((S)-1-{2-[4-(2-Dimethylamino-ethoxy)-phenylamino]...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128958(((S)-3-Methyl-1-{2-[4-(1-methyl-piperidin-4-yloxy)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128954(CHEMBL291587 | {(S)-1-[2-(4-Cyclopentylmethoxy-phe...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128953(CHEMBL64178 | {(S)-1-[2-(4-Isobutoxy-phenylamino)-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128971(CHEMBL304669 | {(S)-1-[2-(4-Cyclohexyloxy-phenylam...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128960(CHEMBL59817 | N-{(S)-1-[2-(4-Benzyloxy-phenylamino...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113674(4-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128952(CHEMBL64367 | {(S)-1-[2-(4-Cyclopropylmethoxy-phen...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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