Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50013359
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29526BDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129625BDBM50129625(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[(5-d...)
Affinity DataKi:  7nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129624BDBM50129624(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[(7-n...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129618BDBM50129618(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[4-(5...)
Affinity DataKi:  24nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129619BDBM50129619(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[8-(5...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129626BDBM50129626(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[3-(5...)
Affinity DataKi:  32nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129621BDBM50129621(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[4-(6...)
Affinity DataKi:  59nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129617BDBM50129617(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(6-am...)
Affinity DataKi:  64nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129628BDBM50129628(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[2-(5...)
Affinity DataKi:  77nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129615BDBM50129615(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[11-(...)
Affinity DataKi:  96nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129622BDBM50129622(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[3-(5...)
Affinity DataKi:  116nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129620BDBM50129620(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[6-(5...)
Affinity DataKi:  180nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129629BDBM50129629(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(6-di...)
Affinity DataKi:  181nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129627BDBM50129627(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[4-(5...)
Affinity DataKi:  183nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129616BDBM50129616(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(5-di...)
Affinity DataKi:  264nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Umr C8076 (Cnrs)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129623BDBM50129623(4-Amino-5-chloro-2-methoxy-benzoic acid 2-{4-[2-(5...)
Affinity DataKi:  1.72E+3nMAssay Description:Binding affinity towards cloned human 5-hydroxytryptamine 4E receptor expressed in C6 glial cells using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed