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Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 50013374
TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11694((2S)-1-[(2S)-2-amino-2-cyclohexylacetyl]pyrrolidin...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards Dipeptidyl peptidase IV (DPP-IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129897(1-(2-Amino-3-methyl-butyryl)-pyrrolidine-2-carboni...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11694((2S)-1-[(2S)-2-amino-2-cyclohexylacetyl]pyrrolidin...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129889(1-[2-(3-Hydroxy-adamantan-1-ylamino)-acetyl]-pyrro...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129889(1-[2-(3-Hydroxy-adamantan-1-ylamino)-acetyl]-pyrro...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) obtained from human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11694((2S)-1-[(2S)-2-amino-2-cyclohexylacetyl]pyrrolidin...)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129945(1-[2-(Adamantan-1-ylamino)-acetyl]-pyrrolidine-2-c...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11694((2S)-1-[(2S)-2-amino-2-cyclohexylacetyl]pyrrolidin...)
Affinity DataIC50:  3.15nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) obtained from human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129889(1-[2-(3-Hydroxy-adamantan-1-ylamino)-acetyl]-pyrro...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129884(6-{4-[2-(2-Cyano-pyrrolidin-1-yl)-2-oxo-ethylamino...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11113(6-{[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP IV) obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11113(6-{[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl...)
Affinity DataIC50:  7nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP IV) obtained from human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129868(1-{2-[4-(5-Trifluoromethyl-pyridin-2-ylamino)-cycl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129865(1-[2-(3-Ethyl-adamantan-1-ylamino)-acetyl]-pyrroli...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50:  8.73nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP IV) obtained from human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129898(1-{2-[4-(Benzothiazol-2-ylamino)-cyclohexylamino]-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129909(1-[2-(Adamantan-2-ylamino)-acetyl]-pyrrolidine-2-c...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129925(1-{2-[4-(4-Chloro-phenoxy)-cyclohexylamino]-acetyl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129912(1-[2-(Bicyclo[2.2.1]hept-2-ylamino)-acetyl]-pyrrol...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129900((1R,2R,3R,5S)1-[2-(2,6,6-Trimethyl-bicyclo[3.1.1]h...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129943(1-[2-(3,5-Dimethyl-adamantan-1-ylamino)-acetyl]-py...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Rat)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50:  17.3nMAssay Description:Inhibitory activity against Dipeptidyl peptidase IV (DPP IV) obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129926(CHEMBL92021 | Cyclohexanecarboxylic acid {4-[2-(2-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM11113(6-{[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129872(CHEMBL319115 | tert-Butyl-carbamic acid 3-[2-(2-cy...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129908(1-[2-(1-Cyclohexanecarbonyl-piperidin-4-ylamino)-a...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129924(1-[2-(1,1-Dimethyl-2-phenyl-ethylamino)-acetyl]-py...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129915(1-[2-(1-Hydroxymethyl-cyclopentylamino)-acetyl]-py...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129902(6-{2-[2-(2-Cyano-pyrrolidin-1-yl)-2-oxo-ethylamino...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129937(1-{2-[2-(Pyridin-2-ylamino)-ethylamino]-acetyl}-py...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM12644((2S)-1-[2-(tert-butylamino)acetyl]pyrrolidine-2-ca...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129940(1-{2-[2-(5-Chloro-pyridin-2-ylamino)-ethylamino]-a...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129881(1-(2-Cyclooctylamino-acetyl)-pyrrolidine-2-carboni...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM12645((2S)-1-[2-(cyclopentylamino)acetyl]pyrrolidine-2-c...)
Affinity DataIC50:  54nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129919(CHEMBL330689 | Phenyl-carbamic acid 3-[2-(2-cyano-...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129932(1-(2-Cycloheptylamino-acetyl)-pyrrolidine-2-carbon...)
Affinity DataIC50:  63nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129907(CHEMBL95093 | Cyclohexyl-carbamic acid 3-[2-(2-cya...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129920(1-(2-Cyclohexylamino-acetyl)-pyrrolidine-2-carboni...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129906(Acetic acid 3-[2-(2-cyano-pyrrolidin-1-yl)-2-oxo-e...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129866(1-(2-Cyclobutylamino-acetyl)-pyrrolidine-2-carboni...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129911(1-{2-[2-(5-Trifluoromethyl-pyridin-2-ylamino)-ethy...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129894(6-{3-[2-(2-Cyano-pyrrolidin-1-yl)-2-oxo-ethylamino...)
Affinity DataIC50:  102nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129935(1-[2-(1-Hydroxymethyl-cyclohexylamino)-acetyl]-pyr...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129882(1-[2-(1,1-Dimethyl-propylamino)-acetyl]-pyrrolidin...)
Affinity DataIC50:  105nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129883(1-[2-(1,1,3,3-Tetramethyl-butylamino)-acetyl]-pyrr...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129888(1-[2-(Indan-2-ylamino)-acetyl]-pyrrolidine-2-carbo...)
Affinity DataIC50:  133nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129901((4-Methoxy-phenyl)-carbamic acid 3-[2-(2-cyano-pyr...)
Affinity DataIC50:  149nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129939(1-{2-[2-(Pyrimidin-2-ylamino)-ethylamino]-acetyl}-...)
Affinity DataIC50:  163nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50129887(CHEMBL274823 | Diisopropyl-carbamic acid 3-[2-(2-c...)
Affinity DataIC50:  183nMAssay Description:Inhibition of human dipeptidyl peptidase IV (DPP IV) obtained from human colonic carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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