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Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50037185
TargetDelta-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027063(CHEMBL2111838)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027063(CHEMBL2111838)
Affinity DataKi:  0.170nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.190nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity determined against Opioid receptor delta 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131967(CHEMBL123898 | N-[2-(5-Phenyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131967(CHEMBL123898 | N-[2-(5-Phenyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131972(4-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.280nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131972(4-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.280nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049807(2-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049807(2-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131968(CHEMBL127828 | Thiophene-3-carboxylic acid {2-[5-(...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.430nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131969(CHEMBL126688 | Thiophene-2-carboxylic acid [2-(5-p...)
Affinity DataKi:  0.450nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131969(CHEMBL126688 | Thiophene-2-carboxylic acid [2-(5-p...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131973(CHEMBL338391 | N-[2-(1-Methyl-5-phenyl-2,3-dihydro...)
Affinity DataKi:  0.470nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131973(CHEMBL338391 | N-[2-(1-Methyl-5-phenyl-2,3-dihydro...)
Affinity DataKi:  0.480nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049806(CHEMBL127969 | Thiophene-2-carboxylic acid [2-(1-m...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049806(CHEMBL127969 | Thiophene-2-carboxylic acid [2-(1-m...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131970(2-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131970(2-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049808(CHEMBL127968 | N-[2-(7-Chloro-1-methyl-5-phenyl-2,...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027062(CHEMBL2111837)
Affinity DataKi:  0.690nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027062(CHEMBL2111837)
Affinity DataKi:  0.690nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027054(CHEMBL2448130)
Affinity DataKi:  0.710nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131968(CHEMBL127828 | Thiophene-3-carboxylic acid {2-[5-(...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027057(CHEMBL2448129)
Affinity DataKi:  0.790nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049807(2-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  1nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027055(CHEMBL2448128)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049801(4-Chloro-N-[2-(7-chloro-1-methyl-5-phenyl-2,3-dihy...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049801(4-Chloro-N-[2-(7-chloro-1-methyl-5-phenyl-2,3-dihy...)
Affinity DataKi:  1.30nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049809(CHEMBL126282 | N-[2-(7-Chloro-1-methyl-5-phenyl-2,...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027063(CHEMBL2111838)
Affinity DataKi:  1.5nMAssay Description:Binding affinity determined against Opioid receptor mu 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131969(CHEMBL126688 | Thiophene-2-carboxylic acid [2-(5-p...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131968(CHEMBL127828 | Thiophene-3-carboxylic acid {2-[5-(...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity of compound was determined against Opioid receptor mu 1 from native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi:  1.90nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027055(CHEMBL2448128)
Affinity DataKi:  2.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3nMAssay Description:Binding affinity of compound was determined against Opioid receptor mu 1 from native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3nMAssay Description:Binding affinity determined against Opioid receptor mu 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131968(CHEMBL127828 | Thiophene-3-carboxylic acid {2-[5-(...)
Affinity DataKi:  3nMAssay Description:Binding affinity determined against Opioid receptor mu 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131966(CHEMBL126596 | Thiophene-2-carboxylic acid [2-(6-m...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131971(CHEMBL338393 | Thiophene-2-carboxylic acid methyl-...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131971(CHEMBL338393 | Thiophene-2-carboxylic acid methyl-...)
Affinity DataKi:  4.40nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50027062(CHEMBL2111837)
Affinity DataKi:  4.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50049808(CHEMBL127968 | N-[2-(7-Chloro-1-methyl-5-phenyl-2,...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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