Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50013645
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132855(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132862(4-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 10nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132856(3-Hydroxy-4-[(4-{[2-((1R,2S,5R)-2-isopropyl-5-meth...)
Affinity DataIC50: 100nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132853(3-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 100nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132862(4-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 380nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined by inhibition of Urokinase-type plasminogen activator using primary assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132853(3-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 400nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132863(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 500nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132874(3-Hydroxy-4-({6-[2-((1R,2S,5R)-2-isopropyl-5-methy...)
Affinity DataIC50: 530nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132881(2-{2-Carbamoyl-6-[(4-{[2-((1R,2S,5R)-2-isopropyl-5...)
Affinity DataIC50: 600nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132871(5-Amino-2-{2-[(4-{[2-((1R,2S,5R)-2-isopropyl-5-met...)
Affinity DataIC50: 700nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132876(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 710nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132860(2-{3-Fluoro-2-[(4-{[2-((1R,2S,5R)-2-isopropyl-5-me...)
Affinity DataIC50: 710nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132870(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 890nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132858(4-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 900nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132855(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 940nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132865(3-Hydroxy-4-({4-[2-((1R,2S,5R)-2-isopropyl-5-methy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132883(4-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132875(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 1.20E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined by inhibition of Urokinase-type plasminogen activator using primary assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132875(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 1.20E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132869(3-Hydroxy-4-[(3-{[2-((1R,2S,5R)-2-isopropyl-5-meth...)
Affinity DataIC50: 1.40E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132850(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 1.40E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132877(2-{3-Fluoro-2-[(4-{[2-((1R,2S,5R)-2-isopropyl-5-me...)
Affinity DataIC50: 1.40E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132856(3-Hydroxy-4-[(4-{[2-((1R,2S,5R)-2-isopropyl-5-meth...)
Affinity DataIC50: 1.40E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined by inhibition of Urokinase-type plasminogen activator using primary assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132879(2-(6-Carboxy-2-hydroxy-4-methoxy-3-methyl-phenoxy)...)
Affinity DataIC50: 1.80E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132852(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 2.20E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132868(2-{2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycl...)
Affinity DataIC50: 2.60E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132851(6-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 2.60E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132873(N-[4-(2-Hydroxy-5-nitro-benzylamino)-benzyl]-2-((1...)
Affinity DataIC50: 2.70E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132878(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 2.90E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132867(1-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50: 2.90E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132857(4-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohe...)
Affinity DataIC50: 3.20E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132864(3-Hydroxy-4-[(4-{2-[2-((1R,2S,5R)-2-isopropyl-5-me...)
Affinity DataIC50: 3.90E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132882(3-Hydroxy-4-{[4-({[2-((1R,2S,5R)-2-isopropyl-5-met...)
Affinity DataIC50: 5.00E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132861(3-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohe...)
Affinity DataIC50: 7.80E+3nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132866(2-[(4-{[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohe...)
Affinity DataIC50: 1.50E+4nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132880(3-Hydroxy-4-{4-[2-((1R,2S,5R)-2-isopropyl-5-methyl...)
Affinity DataIC50: 1.50E+4nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132859(2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexyloxy)-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132872(2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexyloxy)-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132854(N-(4-Benzylamino-benzyl)-2-((1R,2S,5R)-2-isopropyl...)
Affinity DataIC50: 1.50E+4nMAssay Description:Plasminogen Activator Inhibitor-1 (PAI-1) activity was determined using plasma clot lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed