Compile Data Set for Download or QSAR
Report error Found 193 Enz. Inhib. hit(s) with all data for entry = 1847 Sort by
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14593(CHEMBL77076 | 3-amino-5-[1-({[(4-carbamimidoylphen...)
Affinity DataIC50: 16nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14535(2-[6-(3-aminophenyl)-5-chloro-2-oxo-3-(propan-2-yl...)
Affinity DataIC50: 20nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14543(2-[6-(3-aminophenyl)-5-chloro-3-(cyclobutylamino)-...)
Affinity DataIC50: 20nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14528(2-[6-(3-aminophenyl)-5-chloro-3-(ethylamino)-2-oxo...)
Affinity DataIC50: 40nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14519(N-[(4-carbamimidoylphenyl)methyl]-2-(5-chloro-3-{[...)
Affinity DataIC50: 40nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14520(N-[(4-carbamimidoylphenyl)methyl]-2-(5-chloro-3-{[...)
Affinity DataIC50: 40nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14563(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-6-et...)
Affinity DataIC50: 40nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14537(2-[6-(3-aminophenyl)-5-chloro-2-oxo-3-(pentan-3-yl...)
Affinity DataIC50: 50nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14526(2-[6-(3-aminophenyl)-5-chloro-3-(methylamino)-2-ox...)
Affinity DataIC50: 60nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14562(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-6-me...)
Affinity DataIC50: 60nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14583(2-[6-(3-aminophenyl)-5-chloro-2-oxo-3-[(2-phenylet...)
Affinity DataIC50: 70nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14552(2-[6-(3-aminophenyl)-5-chloro-3-[(3-hydroxypropyl)...)
Affinity DataIC50: 90nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14533(2-[6-(3-aminophenyl)-3-(butylamino)-5-chloro-2-oxo...)
Affinity DataIC50: 100nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14571(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(4...)
Affinity DataIC50: 100nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14592(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(3...)
Affinity DataIC50: 100nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14590(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(3...)
Affinity DataIC50: 110nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14550(2-[6-(3-aminophenyl)-5-chloro-3-[(2-methoxyethyl)a...)
Affinity DataIC50: 140nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14501(N-[(6-carbamimidoylpyridin-3-yl)methyl]-2-{2-oxo-6...)
Affinity DataIC50: 150nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14498(CHEMBL75084 | N-[(4-carbamimidoylphenyl)methyl]-2-...)
Affinity DataIC50: 160nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14520(N-[(4-carbamimidoylphenyl)methyl]-2-(5-chloro-3-{[...)
Affinity DataIC50: 180nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14514(CHEMBL78053 | (2R)-N-[(1S)-1-{[(2S)-5-carbamimidam...)
Affinity DataIC50: 200nMpH: 8.0 T: 2°CAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14534(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-ox...)
Affinity DataIC50: 200nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14584(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(c...)
Affinity DataIC50: 200nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14568(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(4...)
Affinity DataIC50: 200nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14499(N-[(4-carbamimidoylphenyl)methyl]-2-{2-oxo-6-pheny...)
Affinity DataIC50: 300nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14575(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(2...)
Affinity DataIC50: 300nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14577(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(4...)
Affinity DataIC50: 300nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14499(N-[(4-carbamimidoylphenyl)methyl]-2-{2-oxo-6-pheny...)
Affinity DataIC50: 340nMpH: 8.0 T: 2°CAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14585(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(c...)
Affinity DataIC50: 340nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14587(3-[1-({[(4-carbamimidoylphenyl)methyl]carbamoyl}me...)
Affinity DataIC50: 360nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14527(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(e...)
Affinity DataIC50: 400nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14529(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-ox...)
Affinity DataIC50: 400nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14542(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(c...)
Affinity DataIC50: 400nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14536(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-ox...)
Affinity DataIC50: 430nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14575(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(2...)
Affinity DataIC50: 430nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14591(N-{3-[1-({[(4-carbamimidoylphenyl)methyl]carbamoyl...)
Affinity DataIC50: 450nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14554(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-3-[(...)
Affinity DataIC50: 470nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14548(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-3-[(...)
Affinity DataIC50: 500nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14551(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-3-[(...)
Affinity DataIC50: 500nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14588(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-6-[3...)
Affinity DataIC50: 580nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14519(N-[(4-carbamimidoylphenyl)methyl]-2-(5-chloro-3-{[...)
Affinity DataIC50: 600nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14553(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-3-[(...)
Affinity DataIC50: 600nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14588(N-[(4-carbamimidoylphenyl)methyl]-2-{5-chloro-6-[3...)
Affinity DataIC50: 600nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14592(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(3...)
Affinity DataIC50: 600nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14498(CHEMBL75084 | N-[(4-carbamimidoylphenyl)methyl]-2-...)
Affinity DataIC50: 630nMpH: 8.0 T: 2°CAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14557(2-[6-(3-aminophenyl)-5-chloro-3-{[2-(dimethylamino...)
Affinity DataIC50: 690nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14525(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(m...)
Affinity DataIC50: 700nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14530(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-ox...)
Affinity DataIC50: 700nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCoagulation factor VII(Human)
Pharmacia

LigandPNGBDBM14531(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-ox...)
Affinity DataIC50: 720nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProthrombin(Human)
Pharmacia

LigandPNGBDBM14567(N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-6-(3...)
Affinity DataIC50: 720nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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