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Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50036059
TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50001561(5-(6-Imino-3-thiophen-3-yl-6H-pyridazin-1-ylmethyl...)
Affinity DataIC50:  88nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50001562(5-(6-Imino-3-phenyl-6H-pyridazin-1-ylmethyl)-isoxa...)
Affinity DataIC50:  240nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50001556(4-(6-Imino-5-methyl-3-phenyl-6H-pyridazin-1-yl)-bu...)
Affinity DataIC50:  800nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed