Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50022503
Affinity DataIC50: 20nMAssay Description:Inhibition of glutathione S-transferase fused Met (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HGF-dependent Met (unknown origin) phosphorylationMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Dana-Farber Cancer Institute
Curated by ChEMBL
Dana-Farber Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of glutathione S-transferase fused Flk1 (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of glutathione S-transferase fused FGFR1 (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of glutathione S-transferase fused CDK2 (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Dana-Farber Cancer Institute
Curated by ChEMBL
Dana-Farber Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of glutathione S-transferase fused c-Src (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Human)
Dana-Farber Cancer Institute
Curated by ChEMBL
Dana-Farber Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of glutathione S-transferase fused PDGFbetaR (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substra...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of glutathione S-transferase fused Tie2 (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of glutathione S-transferase fused EGFR (unknown origin) catalytic activity infected in Sf9 cells using poly-Glu-Tyr (4:1) as substrateMore data for this Ligand-Target Pair
