Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 1173
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9606BDBM9606((2R,3S,4S,5R)-1,6-bis[(2-fluorophenyl)methoxy]-2,5...)
Affinity DataIC50: 200nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9605BDBM9605((2R,3S,4S,5R)-1,6-bis[(2,6-difluorophenyl)methoxy]...)
Affinity DataIC50: 330nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9594BDBM9594((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2,6-difl...)
Affinity DataIC50: 330nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9593BDBM9593((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2-fluoro...)
Affinity DataIC50: 600nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9576BDBM9576((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-fluoro...)
Affinity DataIC50: 700nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9604BDBM9604((2R,3S,4S,5R)-1,6-bis[(2-fluorophenyl)methoxy]-2,5...)
Affinity DataIC50: 800nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9603BDBM9603((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis({[4-(hydr...)
Affinity DataIC50: 1.20E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9592BDBM9592((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(3-fluoro...)
Affinity DataIC50: 1.50E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9574BDBM9574((2R,3S,4S,5R)-1,2,5,6-tetrakis[(4-fluorophenyl)met...)
Affinity DataIC50: 1.60E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9579BDBM9579((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(3-fluoro...)
Affinity DataIC50: 1.80E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9601BDBM9601(tetra-O-benzyl-d-mannitol deriv. 1ee)
Affinity DataIC50: 2.00E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9577BDBM9577((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-chloro...)
Affinity DataIC50: 2.00E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9578BDBM9578((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-bromop...)
Affinity DataIC50: 2.10E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9571BDBM9571((2R,3S,4S,5R)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...)
Affinity DataIC50: 2.40E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9591BDBM9591((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-fluoro...)
Affinity DataIC50: 2.50E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9582BDBM9582((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2,4-difl...)
Affinity DataIC50: 2.60E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9599BDBM9599((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-methyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9575BDBM9575(4-({[(2R,3S,4S,5R)-1,5,6-tris[(4-cyanophenyl)metho...)
Affinity DataIC50: 3.10E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9584BDBM9584((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-methyl...)
Affinity DataIC50: 3.70E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9580BDBM9580((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2-fluoro...)
Affinity DataIC50: 3.70E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9595BDBM9595((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2,4-difl...)
Affinity DataIC50: 4.20E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9600BDBM9600(4-({[(2R,3S,4S,5R)-2,5-bis(benzyloxy)-6-[(4-cyanop...)
Affinity DataIC50: 4.30E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9598BDBM9598((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis({[4-(trif...)
Affinity DataIC50: 5.00E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9602BDBM9602(4-({[(2R,3S,4S,5R)-2,5-bis(benzyloxy)-6-[(4-carbox...)
Affinity DataIC50: 5.00E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9597BDBM9597((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-chloro...)
Affinity DataIC50: 5.20E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9585BDBM9585(4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-cyanop...)
Affinity DataIC50: 5.40E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9573BDBM9573((2R,3S,4S,5R)-1,2,5,6-tetrakis({[4-(trifluoromethy...)
Affinity DataIC50: 6.00E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9596BDBM9596((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-bromop...)
Affinity DataIC50: 6.00E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9581BDBM9581((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2,6-difl...)
Affinity DataIC50: 6.40E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9572BDBM9572((2R,3S,4S,5R)-1,2,5,6-tetrakis[(4-methylphenyl)met...)
Affinity DataIC50: 7.00E+3nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9586BDBM9586(tetra-O-benzyl-d-mannitol deriv. 1p)
Affinity DataIC50: 8.40E+3nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9583BDBM9583((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis({[4-(trif...)
Affinity DataIC50: 1.00E+4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9588BDBM9588((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis({[4-(hydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9590BDBM9590(4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-carbam...)
Affinity DataIC50: 2.00E+4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9587BDBM9587(4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-carbox...)
Affinity DataIC50: 2.60E+4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9589BDBM9589((2R,3S,4S,5R)-2,5-bis({[4-(aminomethyl)phenyl]meth...)
Affinity DataIC50: 2.70E+4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9566BDBM9566((2R,3S,4S,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9567BDBM9567((2R,3R,4S,5R)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9568BDBM9568((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-diphenoxyhexa...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9569BDBM9569((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-diphenylhexan...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9570BDBM9570((2R,3S,5S)-1,2,5,6-tetrakis(benzyloxy)hexan-3-ol |...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9564BDBM9564((2S,3R,4R,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9565BDBM9565((2R,3R,4S,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...)
Affinity DataIC50: 5.00E+4nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2006
Entry Details Article
PubMed