Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 5440
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.0636nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.143nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.151nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.161nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.163nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.172nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.173nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.174nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | Morphine | NSC_5980)
TargetMu-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  1.18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86417(5-amino-2-{1-[1-[1-amino-2-(4-hydroxyphenyl)ethylc...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  1.22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM50060070((S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phe...)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86419(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86415(Tyr-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  2.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  2.83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM50060070((S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phe...)
Affinity DataKi:  3.44nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | Morphine | NSC_5980)
Affinity DataKi:  5.64nMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86417(5-amino-2-{1-[1-[1-amino-2-(4-hydroxyphenyl)ethylc...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86415(Tyr-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  12.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86419(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  213nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  1.67E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed