Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50013816 Sort by
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataIC50: 8.40nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134963(Phosphoric acid mono-[(1R,5S)-4-(2-bromo-6-methyla...)
Affinity DataIC50: 37nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409764(CHEMBL2112867)
Affinity DataIC50: 49nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409757(CHEMBL2112864)
Affinity DataIC50: 52nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134966(Phosphoric acid mono-[(1R,5S)-4-(6-amino-2-iodo-pu...)
Affinity DataIC50: 87nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409761(CHEMBL2112863)
Affinity DataIC50: 157nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409762(CHEMBL2112865)
Affinity DataIC50: 221nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409759(CHEMBL2112868)
Affinity DataIC50: 356nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409760(CHEMBL2112861)
Affinity DataIC50: 367nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134967(Phosphoric acid mono-[(1R,5S)-4-(6-methylamino-2-m...)
Affinity DataIC50: 377nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409758(CHEMBL2112869)
Affinity DataIC50: 452nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409756(CHEMBL2112866)
Affinity DataIC50: 1.87E+3nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409763(CHEMBL2112007)
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataKi:  0.780nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409757(CHEMBL2112864)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409764(CHEMBL2112867)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134963(Phosphoric acid mono-[(1R,5S)-4-(2-bromo-6-methyla...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134966(Phosphoric acid mono-[(1R,5S)-4-(6-amino-2-iodo-pu...)
Affinity DataKi:  12.6nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409761(CHEMBL2112863)
Affinity DataKi:  17.6nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50134967(Phosphoric acid mono-[(1R,5S)-4-(6-methylamino-2-m...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409759(CHEMBL2112868)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409758(CHEMBL2112869)
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409762(CHEMBL2112865)
Affinity DataKi:  91nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409756(CHEMBL2112866)
Affinity DataKi:  330nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409763(CHEMBL2112007)
Affinity DataKi:  430nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 1(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50409760(CHEMBL2112861)
Affinity DataKi:  863nMAssay Description:Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed