Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50035339 Sort by
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50135425(4-{2-(Isoquinoline-5-sulfonylamino)-3-[4-(isoquino...)
Affinity DataIC50: 1nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50087267((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataIC50: 51nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50414329(CHEMBL336545)
Affinity DataIC50: 158nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50421620(CHEMBL337984)
Affinity DataIC50: 398nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50414328(CHEMBL339140)
Affinity DataIC50: 501nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50421619(CHEMBL339145)
Affinity DataIC50: 3.98E+3nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 7(Human)
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50414319(CHEMBL128907)
Affinity DataIC50: 3.98E+3nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed