Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 5447
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(NSC_105100 | CAS_105100 | 12-Deoxyphorbol 13-pheny...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(NSC_4179 | CAS_4179 | Mezerein)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(NSC_105100 | CAS_105100 | 12-Deoxyphorbol 13-pheny...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(NSC_4179 | CAS_4179 | Mezerein)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432(CAS_159320 | NSC_159320 | (-)-Octylindolactam V)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432(CAS_159320 | NSC_159320 | (-)-Octylindolactam V)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(NSC_4179 | CAS_4179 | Mezerein)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(NSC_105100 | CAS_105100 | 12-Deoxyphorbol 13-pheny...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432(CAS_159320 | NSC_159320 | (-)-Octylindolactam V)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  3.57nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  3.85nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  4.83nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V (low PS) | NSC_105000 | CAS_10500...)
Affinity DataKi:  8.16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(NSC_6437389 | CAS_6437389 | Thymeleatoxin (low PS)...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  11.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V (low PS) | NSC_105000 | CAS_10500...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  24.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 (low PS) | B8-DL-B8)
Affinity DataKi:  26.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  28.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V (low PS) | NSC_105000 | CAS_10500...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V (low PS) | NSC_105000 | CAS_10500...)
Affinity DataKi:  43.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V (low PS) | NSC_105000 | CAS_10500...)
Affinity DataKi:  48.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetPolycystin-1(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(NSC_104731 | CAS_104731 | OAG)
Affinity DataKi:  146nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(NSC_104731 | CAS_104731 | OAG)
Affinity DataKi:  224nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(NSC_104731 | CAS_104731 | OAG)
Affinity DataKi:  230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed