Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 5447
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  3.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  4.83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  8.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  11.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  24.6nMMore data for this Ligand-Target Pair
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  26.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  28.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  43.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  48.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  146nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  224nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed