Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50036074
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368463BDBM50368463(CHEMBL608175)
Affinity DataEC50:  832nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368472BDBM50368472(CHEMBL611920)
Affinity DataEC50:  2.63E+3nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368485BDBM50368485(CHEMBL611609)
Affinity DataEC50:  3.02E+3nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368471BDBM50368471(CHEMBL608174)
Affinity DataEC50:  4.17E+3nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368480BDBM50368480(CHEMBL607590)
Affinity DataEC50:  8.91E+3nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368487BDBM50368487(CHEMBL607508)
Affinity DataEC50:  9.12E+3nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368467BDBM50368467(CHEMBL607886)
Affinity DataEC50:  1.20E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368474BDBM50368474(CHEMBL608167)
Affinity DataEC50:  1.23E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368466BDBM50368466(CHEMBL611947)
Affinity DataEC50:  1.26E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368475BDBM50368475(CHEMBL608745)
Affinity DataEC50:  1.41E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368468BDBM50368468(CHEMBL607511)
Affinity DataEC50:  1.70E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368484BDBM50368484(CHEMBL607872)
Affinity DataEC50:  1.91E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368465BDBM50368465(CHEMBL608451)
Affinity DataEC50:  1.95E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368478BDBM50368478(CHEMBL610444)
Affinity DataEC50:  2.00E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368488BDBM50368488(CHEMBL611610)
Affinity DataEC50:  2.29E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368492BDBM50368492(CHEMBL607798)
Affinity DataEC50:  2.63E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368481BDBM50368481(CHEMBL607604)
Affinity DataEC50:  3.09E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368482BDBM50368482(CHEMBL608447)
Affinity DataEC50:  3.24E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368489BDBM50368489(CHEMBL611571)
Affinity DataEC50:  3.98E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368479BDBM50368479(CHEMBL611918)
Affinity DataEC50:  4.17E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368476BDBM50368476(CHEMBL608448)
Affinity DataEC50:  4.17E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368464BDBM50368464(CHEMBL608176)
Affinity DataEC50:  4.17E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368486BDBM50368486(CHEMBL608668)
Affinity DataEC50:  4.37E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368483BDBM50368483(CHEMBL607605)
Affinity DataEC50:  4.90E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368469BDBM50368469(CHEMBL609338)
Affinity DataEC50:  4.90E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368473BDBM50368473(CHEMBL607797)
Affinity DataEC50:  5.75E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368491BDBM50368491(CHEMBL610445)
Affinity DataEC50:  6.03E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368470BDBM50368470(CHEMBL607891)
Affinity DataEC50:  6.61E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368477BDBM50368477(CHEMBL607592)
Affinity DataEC50:  8.32E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368490BDBM50368490(CHEMBL607874)
Affinity DataEC50:  8.32E+4nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
University of South Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009530BDBM50009530(CHEMBL88070 | 3-(4-{2-[6-Amino-9-(3,4-dihydroxy-5-...)
Affinity DataEC50:  1.12E+5nMAssay Description:Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed