Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50000295
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 83449BDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataKi:  65nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004109BDBM50004109(CHEMBL142577 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  582nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004111BDBM50004111(CHEMBL343429 | 1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  644nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004113BDBM50004113(CHEMBL347761 | 1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  711nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 83449BDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataKi:  1.09E+3nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004112BDBM50004112(CHEMBL358455 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  1.13E+3nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004113BDBM50004113(CHEMBL347761 | 1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  3.72E+3nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004109BDBM50004109(CHEMBL142577 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  4.45E+3nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004110BDBM50004110(CHEMBL356855 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  7.28E+3nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004112BDBM50004112(CHEMBL358455 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  8.22E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004111BDBM50004111(CHEMBL343429 | 1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)...)
Affinity DataKi:  1.63E+4nMAssay Description:Compound was evaluated for its ability to displace [3H](+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004110BDBM50004110(CHEMBL356855 | 1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)...)
Affinity DataKi:  2.90E+4nMAssay Description:Compound was evaluated for its ability to displace [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed