Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50014149
Displayed 1 to 50 (of 72 total ) | Next | Last >>
Affinity DataKi: 3nMAssay Description:Binding affinity towards metabotropic glutamate receptor 3 was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity towards metabotropic glutamate receptor 2 was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 147nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.32E+3nMAssay Description:Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 8.80E+3nMAssay Description:Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Metabotropic glutamate receptor 3 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards metabotropic glutamate receptor 2 was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+4nMAssay Description:Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+4nMAssay Description:Metabotropic glutamate receptor 1 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+4nMAssay Description:Metabotropic glutamate receptor 4 antagonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+4nMAssay Description:Metabotropic glutamate receptor 8 antagonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+4nMAssay Description:Metabotropic glutamate receptor 1 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+4nMAssay Description:Metabotropic glutamate receptor 6 antagonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+4nMAssay Description:Metabotropic glutamate receptor 7 antagonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+4nMAssay Description:Metabotropic glutamate receptor 7 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 1 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 1 agonist activity as basal [3H]- IP formation in ratMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 7 agonist activity to influence forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat non neuronal cellsMore data for this Ligand-Target Pair



3D Structure (crystal)






