Compile Data Set for Download or QSAR
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Found 34 Enz. Inhib. hit(s) with all data for entry = 50014211
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50132862(4-{3-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cyclohexy...)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139534(2-[2-Methoxy-6-({3-trifluoromethyl-4-[4-(3-trifluo...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139536(1-[3-Fluoro-6-nitro-2-({3-trifluoromethyl-4-[4-(3-...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139540(5-Bromo-2-[3-fluoro-2-({3-trifluoromethyl-4-[4-(3-...)
Affinity DataIC50:  800nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139562(1-{2-Nitro-4-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  880nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139546(6-[2-Methoxy-6-({3-trifluoromethyl-4-[4-(3-trifluo...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139532(5-Chloro-2-[2-methoxy-6-({3-trifluoromethyl-4-[4-(...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139548(3-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139542(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  910nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139561(1-[3-Fluoro-2-({3-trifluoromethyl-4-[4-(3-trifluor...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139541(2-[4-Nitro-2-({3-trifluoromethyl-4-[4-(3-trifluoro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139564(1-{4-Nitro-2-trifluoromethyl-5-[4-(4-trifluorometh...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139556(4-({2,4-Dinitro-5-[4-(3-trifluoromethyl-phenyl)-pi...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139552(1-[3-Fluoro-6-nitro-2-({3-trifluoromethyl-4-[4-(3-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139537(4-({4-Nitro-2-trifluoromethyl-5-[4-(3-trifluoromet...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139559(1-[3-Fluoro-2-({3-trifluoromethyl-4-[4-(3-trifluor...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139549(1-[3-Trifluoromethyl-2-({3-trifluoromethyl-4-[4-(3...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139563(4-({3-Trifluoromethyl-4-[4-(3-trifluoromethyl-phen...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139545(({2-Nitro-4-trifluoromethyl-5-[4-(3-trifluoromethy...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139555(4-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139554(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139538(4-({2-Nitro-5-[4-(3-trifluoromethyl-phenyl)-pipera...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139543(1-{4-Nitro-2-trifluoromethyl-5-[4-(5-trifluorometh...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139551(4-({3-Nitro-6-[4-(3-trifluoromethyl-phenyl)-pipera...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139533(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139550(3-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139535(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139539(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139547(4-({5-Nitro-6-[4-(3-trifluoromethyl-phenyl)-pipera...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139553(4-({4-Nitro-3-[4-(3-trifluoromethyl-phenyl)-pipera...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139558(1-{4-Nitro-2-trifluoromethyl-5-[4-(3-trifluorometh...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139560(1-(5-{4-[2-((1R,2S,5R)-2-Isopropyl-5-methyl-cycloh...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139557(6-(4-Carboxy-benzylamino)-3-nitro-2-[4-(3-trifluor...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50139544(1-{5-[4-(2,6-Dinitro-3-trifluoromethyl-phenyl)-pip...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibitory concentration against plasminogen activator inhibitor-1 (PAI-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed