Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 798
LigandChemical structure of BindingDB Monomer ID 6204BDBM6204(N-(3-chloro-1-benzofuran-7-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6219BDBM6219(BMCL182776 Compound 1 | N-(5-chloro-2H-1,3-benzodi...)
Affinity DataIC50: 4nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6210BDBM6210(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-6-methoxy-7-[...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6211BDBM6211(N-(5-Bromo-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-mo...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6218BDBM6218(AZD0530 analogue 34 | N-(5-chloro-2H-1,3-benzodiox...)
Affinity DataIC50: 5nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6202BDBM6202(N-(6-chloro-1-benzofuran-7-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6220BDBM6220(4-[({4-[(5-chloro-2H-1,3-benzodioxol-4-yl)amino]-6...)
Affinity DataIC50: 10nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6196BDBM6196(N-(2-Chloro-5-methoxyphenyl)-6-methoxy-7-(3-morpho...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6198BDBM6198(AZD0530 analogue 35 | M475271 | N-(2-Chloro-5-meth...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6200BDBM6200(N-(5-chloro-1-benzofuran-4-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6216BDBM6216(N-(5-Chloro-1,3-benzodioxol-4-yl)-7-(3-morpholin-4...)
Affinity DataIC50: 10nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6209BDBM6209(N-(2H-1,3-benzodioxol-4-yl)-6-methoxy-7-[3-(morpho...)
Affinity DataIC50: 14nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6199BDBM6199(N-(1-benzofuran-4-yl)-6-methoxy-7-[3-(morpholin-4-...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6208BDBM6208(N-(3-chloro-1H-indol-7-yl)-6-methoxy-7-[3-(morphol...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6212BDBM6212(N-(5-Fluoro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-m...)
Affinity DataIC50: 28nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6201BDBM6201(N-(1-benzofuran-7-yl)-6-methoxy-7-[3-(morpholin-4-...)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6193BDBM6193(6-Methoxy-N-(3-methoxyphenyl)-7-(3-morpholin-4-ylp...)
Affinity DataIC50: 37nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6206BDBM6206(6-methoxy-N-(1-methyl-1H-indol-4-yl)-7-[3-(morphol...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6217BDBM6217(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-methoxy-6-[...)
Affinity DataIC50: 50nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6204BDBM6204(N-(3-chloro-1-benzofuran-7-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 100nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6205BDBM6205(N-(1H-indol-4-yl)-6-methoxy-7-(3-morpholin-4-ylpro...)
Affinity DataIC50: 177nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6199BDBM6199(N-(1-benzofuran-4-yl)-6-methoxy-7-[3-(morpholin-4-...)
Affinity DataIC50: 250nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 4394BDBM4394(6,7-dimethoxy-N-(3-methoxyphenyl)quinazolin-4-amin...)
Affinity DataIC50: 253nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6207BDBM6207(N-(1H-indol-7-yl)-6-methoxy-7-(3-morpholin-4-ylpro...)
Affinity DataIC50: 260nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6213BDBM6213(N-(2,2-Difluoro-1,3-benzodioxol-4-yl)-6-methoxy-7-...)
Affinity DataIC50: 270nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6215BDBM6215(N-(2,3-dihydro-1,4-benzodioxin-5-yl)-6-methoxy-7-[...)
Affinity DataIC50: 370nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6201BDBM6201(N-(1-benzofuran-7-yl)-6-methoxy-7-[3-(morpholin-4-...)
Affinity DataIC50: 410nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6206BDBM6206(6-methoxy-N-(1-methyl-1H-indol-4-yl)-7-[3-(morphol...)
Affinity DataIC50: 420nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6203BDBM6203(N-(2,3-dihydro-1-benzofuran-7-yl)-6-methoxy-7-[3-(...)
Affinity DataIC50: 433nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6195BDBM6195(6-Methoxy-N-(4-methoxyphenyl)-7-(3-morpholin-4-ylp...)
Affinity DataIC50: 477nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6194BDBM6194(6-methoxy-N-(2-methoxyphenyl)-7-[3-(morpholin-4-yl...)
Affinity DataIC50: 560nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6198BDBM6198(AZD0530 analogue 35 | M475271 | N-(2-Chloro-5-meth...)
Affinity DataIC50: 670nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6214BDBM6214(N-(1,3-Benzodioxol-5-yl)-6-methoxy-7-(3-morpholin-...)
Affinity DataIC50: 760nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6197BDBM6197(N-(2-Chloro-5-ethoxyphenyl)-6-methoxy-7-(3-morphol...)
Affinity DataIC50: 963nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6193BDBM6193(6-Methoxy-N-(3-methoxyphenyl)-7-(3-morpholin-4-ylp...)
Affinity DataIC50: 1.11E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6196BDBM6196(N-(2-Chloro-5-methoxyphenyl)-6-methoxy-7-(3-morpho...)
Affinity DataIC50: 1.18E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6200BDBM6200(N-(5-chloro-1-benzofuran-4-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 1.23E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6202BDBM6202(N-(6-chloro-1-benzofuran-7-yl)-6-methoxy-7-[3-(mor...)
Affinity DataIC50: 1.38E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6208BDBM6208(N-(3-chloro-1H-indol-7-yl)-6-methoxy-7-[3-(morphol...)
Affinity DataIC50: 2.32E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6209BDBM6209(N-(2H-1,3-benzodioxol-4-yl)-6-methoxy-7-[3-(morpho...)
Affinity DataIC50: 4.96E+3nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6212BDBM6212(N-(5-Fluoro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-m...)
Affinity DataIC50: 8.16E+3nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6218BDBM6218(AZD0530 analogue 34 | N-(5-chloro-2H-1,3-benzodiox...)
Affinity DataIC50: 1.56E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6210BDBM6210(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-6-methoxy-7-[...)
Affinity DataIC50: 1.70E+4nMT: 2°CAssay Description:An ELISA assay was used to determine the ability of inhibitor to inhibit VEGF-RRTK activity. The compounds were incubated with enzyme 20 min at room ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6219BDBM6219(BMCL182776 Compound 1 | N-(5-chloro-2H-1,3-benzodi...)
Affinity DataIC50: 2.17E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6211BDBM6211(N-(5-Bromo-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-mo...)
Affinity DataIC50: 4.26E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6217BDBM6217(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-methoxy-6-[...)
Affinity DataIC50: 7.38E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6220BDBM6220(4-[({4-[(5-chloro-2H-1,3-benzodioxol-4-yl)amino]-6...)
Affinity DataIC50: 7.70E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6216BDBM6216(N-(5-Chloro-1,3-benzodioxol-4-yl)-7-(3-morpholin-4...)
Affinity DataIC50: 9.14E+4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6218BDBM6218(AZD0530 analogue 34 | N-(5-chloro-2H-1,3-benzodiox...)
Affinity DataIC50: 1.00E+5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6219BDBM6219(BMCL182776 Compound 1 | N-(5-chloro-2H-1,3-benzodi...)
Affinity DataIC50: 1.00E+5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2005
Entry Details Article
PubMed
Displayed 1 to 50 (of 54 total ) | Next | Last >>
Jump to: