Affinity DataKi: 2.60nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-ZM-241,385 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 11.8nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-ZM-241,385 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 18.9nMAssay Description:Binding affinity for human HEK-293 adenosine A2B receptor using [125I]-ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 53.4nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-ZM-241,385 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-ZM-241,385 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 183nMAssay Description:Binding affinity for human adenosine A3 receptor using [3H]-PBS-11 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 415nMAssay Description:Binding affinity for human HEK-293 adenosine A2B receptor using [125I]-ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 475nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 642nMAssay Description:Displacement of [3H]-MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Dispalcement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+3nMAssay Description:Binding affinity for human HEK-293 adenosine A2B receptor using [125I]-ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]-PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity for human adenosine A3 receptor using [3H]-PBS-11 in CHO cell membranesMore data for this Ligand-Target Pair