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Found 88 Enz. Inhib. hit(s) with all data for entry = 50014299
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140533(CHEMBL25211 | N-[4-((S)-1-Amino-2-oxo-2-thiazolidi...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140529(CHEMBL423108 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-p...)
Affinity DataKi:  5.30E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140535(CHEMBL281178 | N-{4-[(S)-1-Amino-2-((S)-3-fluoro-p...)
Affinity DataKi:  5.50E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140538(CHEMBL23979 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidin...)
Affinity DataKi:  5.70E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140523(CHEMBL22359 | N-[4-((S)-1-Amino-2-oxo-2-thiazolidi...)
Affinity DataKi:  5.90E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140525(CHEMBL281561 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-p...)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140516(CHEMBL23110 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-py...)
Affinity DataKi:  1.60E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140513(CHEMBL23660 | N-{4-[(S)-1-Amino-2-((S)-3-fluoro-py...)
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140536((S)-2-Amino-2-cyclohexyl-1-thiazolidin-3-yl-ethano...)
Affinity DataKi:  2.80E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140526(CHEMBL278558 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidi...)
Affinity DataKi:  2.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140521(CHEMBL25437 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidin...)
Affinity DataKi:  3.50E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140512(CHEMBL23891 | {4-[(S)-1-Amino-2-((S)-3-fluoro-pyrr...)
Affinity DataKi:  3.70E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140517(CHEMBL283368 | N-[4-((S)-1-Amino-2-oxo-2-thiazolid...)
Affinity DataKi:  3.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140515(CHEMBL22679 | [4-((S)-1-Amino-2-oxo-2-pyrrolidin-1...)
Affinity DataKi:  4.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140518(CHEMBL279944 | {4-[(S)-1-Amino-2-(3,3-difluoro-pyr...)
Affinity DataKi:  4.20E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140531(CHEMBL277693 | {4-[(S)-1-Amino-2-((R)-3-fluoro-pyr...)
Affinity DataKi:  4.30E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11463(CHEMBL22310 | N-{4-[(1S)-1-amino-2-[(3S)-3-fluorop...)
Affinity DataKi:  4.90E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140522(CHEMBL283309 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-p...)
Affinity DataKi:  5.20E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140524(CHEMBL23924 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-py...)
Affinity DataKi:  7.30E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140539((S)-2-Amino-2-cyclohexyl-1-((R)-3-fluoro-pyrrolidi...)
Affinity DataKi: >9.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140527((S)-2-Amino-2-cyclohexyl-1-((S)-3-fluoro-pyrrolidi...)
Affinity DataKi: >9.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140541((S)-2-Amino-2-cyclohexyl-1-(3,3-difluoro-pyrrolidi...)
Affinity DataKi: >9.00E+4nMAssay Description:Binding affinity of the compound towards human ERG potassium ion channel was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140530(CHEMBL22294 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-py...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140533(CHEMBL25211 | N-[4-((S)-1-Amino-2-oxo-2-thiazolidi...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140529(CHEMBL423108 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-p...)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140520(CHEMBL23176 | [4-((S)-1-Amino-2-oxo-2-thiazolidin-...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140518(CHEMBL279944 | {4-[(S)-1-Amino-2-(3,3-difluoro-pyr...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140535(CHEMBL281178 | N-{4-[(S)-1-Amino-2-((S)-3-fluoro-p...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11463(CHEMBL22310 | N-{4-[(1S)-1-amino-2-[(3S)-3-fluorop...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140523(CHEMBL22359 | N-[4-((S)-1-Amino-2-oxo-2-thiazolidi...)
Affinity DataIC50:  53nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140513(CHEMBL23660 | N-{4-[(S)-1-Amino-2-((S)-3-fluoro-py...)
Affinity DataIC50:  54nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140516(CHEMBL23110 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-py...)
Affinity DataIC50:  55nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140512(CHEMBL23891 | {4-[(S)-1-Amino-2-((S)-3-fluoro-pyrr...)
Affinity DataIC50:  56nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140522(CHEMBL283309 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-p...)
Affinity DataIC50:  58nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140517(CHEMBL283368 | N-[4-((S)-1-Amino-2-oxo-2-thiazolid...)
Affinity DataIC50:  67nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140528(CHEMBL277635 | N-{4-[(S)-1-Amino-2-(3,3-difluoro-p...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140541((S)-2-Amino-2-cyclohexyl-1-(3,3-difluoro-pyrrolidi...)
Affinity DataIC50:  73nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140525(CHEMBL281561 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-p...)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140521(CHEMBL25437 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidin...)
Affinity DataIC50:  88nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140531(CHEMBL277693 | {4-[(S)-1-Amino-2-((R)-3-fluoro-pyr...)
Affinity DataIC50:  88nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140536((S)-2-Amino-2-cyclohexyl-1-thiazolidin-3-yl-ethano...)
Affinity DataIC50:  89nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140538(CHEMBL23979 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidin...)
Affinity DataIC50:  89nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140515(CHEMBL22679 | [4-((S)-1-Amino-2-oxo-2-pyrrolidin-1...)
Affinity DataIC50:  94nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140524(CHEMBL23924 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-py...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140527((S)-2-Amino-2-cyclohexyl-1-((S)-3-fluoro-pyrrolidi...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140526(CHEMBL278558 | N-[4-((S)-1-Amino-2-oxo-2-pyrrolidi...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140537(CHEMBL23880 | N-{4-[(S)-1-Amino-2-((S)-3-fluoro-py...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140514(CHEMBL23879 | N-{4-[(S)-1-Amino-2-((R)-3-fluoro-py...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140542(CHEMBL277193 | N-{4-[(S)-1-Amino-2-((3R,4R)-3,4-di...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140540(CHEMBL23051 | N-{4-[(S)-1-Amino-2-((3R,4R)-3,4-dif...)
Affinity DataIC50:  270nMAssay Description:Inhibitory activity against human Dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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