Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 2186 Sort by
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17869((3S)-3-amino-1-(cyclopropylamino)heptane-2,2-diol ...)
Affinity DataIC50: 7.00E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17868((2S)-2-amino-4-(methylsulfanyl)-1-(pyridin-2-yl)bu...)
Affinity DataIC50: 1.60E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Morphochem

LigandPNGBDBM17867((2S)-2-amino-4-(methylsulfanyl)-1-(1,3-thiazol-2-y...)
Affinity DataIC50: 1.90E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed