Found 1 Enz. Inhib. hit(s) with all data for entry = 50042086 TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
St. Jude Children'S Research Hospital
Curated by ChEMBL
St. Jude Children'S Research Hospital
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:TP_TRANSPORTER: drug resistance(Imatinib mesylate) in BCRP-expressing SaoS2 cellsMore data for this Ligand-Target Pair
3D Structure (crystal)