Compile Data Set for Download or QSAR
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Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50014559
TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144467(CHEMBL70381 | N-{3-[Benzyl-(4-chloro-2-fluoro-benz...)
Affinity DataIC50:  5.70nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144481(CHEMBL304102 | N-(3-Dibenzylamino-2-ethyl-phenyl)-...)
Affinity DataIC50:  12nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144468(CHEMBL71450 | N-{3-[(4-Allyloxy-benzyl)-benzyl-ami...)
Affinity DataIC50:  13nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144478(CHEMBL420001 | N-{3-[Benzyl-(2-fluoro-benzyl)-amin...)
Affinity DataIC50:  14nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  15nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144488(CHEMBL308743 | N-{3-[Benzyl-(4-chloro-benzyl)-amin...)
Affinity DataIC50:  17nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144456(CHEMBL72182 | N-(5-Benzyl-5,6-dihydro-phenanthridi...)
Affinity DataIC50:  20nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  28nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144493(CHEMBL302248 | N-{3-[Benzyl-(2-chloro-benzyl)-amin...)
Affinity DataIC50:  36nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144480(CHEMBL306697 | N-{3-[Benzyl-(3-fluoro-benzyl)-amin...)
Affinity DataIC50:  42nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144459(CHEMBL68804 | N-{3-[Benzyl-(4-fluoro-benzyl)-amino...)
Affinity DataIC50:  47nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144466(CHEMBL302250 | N-{3-[Benzyl-(2-methyl-benzyl)-amin...)
Affinity DataIC50:  48nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144463(CHEMBL71871 | N-(3-Dibenzylamino-2-hydroxymethyl-p...)
Affinity DataIC50:  56nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144475(CHEMBL70574 | N-{3-[Benzyl-(4-methyl-benzyl)-amino...)
Affinity DataIC50:  58nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144476(CHEMBL302758 | N-{3-[Benzyl-(2-cyano-benzyl)-amino...)
Affinity DataIC50:  60nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144494(CHEMBL71870 | N-{3-[Benzyl-(2-bromo-benzyl)-amino]...)
Affinity DataIC50:  96nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144472(CHEMBL70249 | N-{3-[Benzyl-(4-methoxy-benzyl)-amin...)
Affinity DataIC50:  100nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  100nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144483(CHEMBL305417 | N-{3-[Benzyl-(3-methyl-benzyl)-amin...)
Affinity DataIC50:  110nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144487(CHEMBL304839 | N-{3-[Benzyl-(3-trifluoromethyl-ben...)
Affinity DataIC50:  130nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144477(CHEMBL71818 | Ethanesulfonic acid (3-dibenzylamino...)
Affinity DataIC50:  138nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144478(CHEMBL420001 | N-{3-[Benzyl-(2-fluoro-benzyl)-amin...)
Affinity DataIC50:  150nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144472(CHEMBL70249 | N-{3-[Benzyl-(4-methoxy-benzyl)-amin...)
Affinity DataIC50:  160nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAndrogen receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]-dexamethasone from human androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144467(CHEMBL70381 | N-{3-[Benzyl-(4-chloro-2-fluoro-benz...)
Affinity DataIC50:  210nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144465(CHEMBL70449 | N-{3-[Benzyl-(2-trifluoromethyl-benz...)
Affinity DataIC50:  220nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144461(CHEMBL302134 | N-{3-[Benzyl-(3-trifluoromethoxy-be...)
Affinity DataIC50:  220nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144464(CHEMBL306689 | N-{3-[Benzyl-(3-chloro-benzyl)-amin...)
Affinity DataIC50:  230nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144459(CHEMBL68804 | N-{3-[Benzyl-(4-fluoro-benzyl)-amino...)
Affinity DataIC50:  240nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144470(CHEMBL306491 | N-{3-[Benzyl-(3-methoxy-benzyl)-ami...)
Affinity DataIC50:  250nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  250nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144480(CHEMBL306697 | N-{3-[Benzyl-(3-fluoro-benzyl)-amin...)
Affinity DataIC50:  260nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144481(CHEMBL304102 | N-(3-Dibenzylamino-2-ethyl-phenyl)-...)
Affinity DataIC50:  270nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144482(CHEMBL302580 | N-(3-Dibenzylamino-2-ethoxymethyl-p...)
Affinity DataIC50:  290nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144488(CHEMBL308743 | N-{3-[Benzyl-(4-chloro-benzyl)-amin...)
Affinity DataIC50:  300nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAndrogen receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144467(CHEMBL70381 | N-{3-[Benzyl-(4-chloro-2-fluoro-benz...)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]-dexamethasone from human androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMineralocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]-dexamethasone from human mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144492(CHEMBL304843 | Propane-2-sulfonic acid (3-dibenzyl...)
Affinity DataIC50:  320nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144468(CHEMBL71450 | N-{3-[(4-Allyloxy-benzyl)-benzyl-ami...)
Affinity DataIC50:  340nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144469(CHEMBL69389 | N-{3-[Benzyl-(4-trifluoromethyl-benz...)
Affinity DataIC50:  370nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144477(CHEMBL71818 | Ethanesulfonic acid (3-dibenzylamino...)
Affinity DataIC50:  400nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144470(CHEMBL306491 | N-{3-[Benzyl-(3-methoxy-benzyl)-ami...)
Affinity DataIC50:  450nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144497(CHEMBL71405 | N-(6-Dibenzylamino-biphenyl-2-yl)-me...)
Affinity DataIC50:  450nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144474(4-{[Benzyl-(3-methanesulfonylamino-2-methyl-phenyl...)
Affinity DataIC50:  470nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144498(CHEMBL308204 | N-{3-[Benzyl-(3-cyano-benzyl)-amino...)
Affinity DataIC50:  570nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144494(CHEMBL71870 | N-{3-[Benzyl-(2-bromo-benzyl)-amino]...)
Affinity DataIC50:  580nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144496(CHEMBL72537 | N-(2-Acetyl-3-dibenzylamino-phenyl)-...)
Affinity DataIC50:  580nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144485(CHEMBL71968 | N-{3-[Benzyl-(2-methoxy-benzyl)-amin...)
Affinity DataIC50:  690nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144483(CHEMBL305417 | N-{3-[Benzyl-(3-methyl-benzyl)-amin...)
Affinity DataIC50:  700nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProgesterone receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144467(CHEMBL70381 | N-{3-[Benzyl-(4-chloro-2-fluoro-benz...)
Affinity DataIC50:  790nMAssay Description:Displacement of [3H]-dexamethasone from human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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