Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 971
LigandChemical structure of BindingDB Monomer ID 7665BDBM7665(4-[(5-bromo-4-{imidazo[1,2-a]pyridin-3-yl}pyrimidi...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7655BDBM7655(4-{imidazo[1,2-a]pyridin-3-yl}-N-phenylpyrimidin-2...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7657BDBM7657(CHEMBL73303 | 4-[(4-{imidazo[1,2-a]pyridin-3-yl}py...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7658BDBM7658(4-[(4-{imidazo[1,2-a]pyridin-3-yl}pyrimidin-2-yl)a...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7662BDBM7662(N-[3-(dimethylamino)propyl]-4-[(4-{imidazo[1,2-a]p...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7664BDBM7664(4-[(5-chloro-4-{imidazo[1,2-a]pyridin-3-yl}pyrimid...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7660BDBM7660(4-[(4-{imidazo[1,2-a]pyridin-3-yl}pyrimidin-2-yl)a...)
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7656BDBM7656(N-(3-chlorophenyl)-4-{imidazo[1,2-a]pyridin-3-yl}p...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7661BDBM7661(N-[2-(dimethylamino)ethyl]-4-[(4-{imidazo[1,2-a]py...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7663BDBM7663(N-[3-(dimethylamino)propyl]-4-[(4-{imidazo[1,2-a]p...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7659BDBM7659(CHEMBL309573 | 4-[(4-{imidazo[1,2-a]pyridin-3-yl}p...)
Affinity DataIC50: 12nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7652BDBM7652(N-(3-chlorophenyl)-4-{2-methylimidazo[1,2-a]pyridi...)
Affinity DataIC50: 150nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7661BDBM7661(N-[2-(dimethylamino)ethyl]-4-[(4-{imidazo[1,2-a]py...)
Affinity DataIC50: 260nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7653BDBM7653(N-(4-chlorophenyl)-4-{2-methylimidazo[1,2-a]pyridi...)
Affinity DataIC50: 620nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5374BDBM5374(4-(1H-1,3-benzodiazol-1-yl)-N-(3-chlorophenyl)pyri...)
Affinity DataIC50: 680nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7660BDBM7660(4-[(4-{imidazo[1,2-a]pyridin-3-yl}pyrimidin-2-yl)a...)
Affinity DataIC50: 3.10E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7651BDBM7651(N-(2-chlorophenyl)-4-{2-methylimidazo[1,2-a]pyridi...)
Affinity DataIC50: 8.80E+3nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/13/2006
Entry Details Article
PubMed