Compile Data Set for Download or QSAR
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Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50014660
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  57nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  61nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145690(CHEMBL80977 | {1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity of the compound was tested against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145687(CHEMBL80680 | [(S)-[(S)-2-((R)-2-Benzyloxycarbonyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145693(CHEMBL430813 | [[(S)-2-((R)-2-Benzyloxycarbonylami...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145691(CHEMBL310235 | {1-[(S)-2-((R)-2-Benzyloxycarbonyla...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145692(CHEMBL421318 | [[(S)-2-((R)-2-Benzyloxycarbonylami...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibitory activity of the compound was tested against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTissue-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity of the compound was tested against Tissue type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory activity of the compound was tested against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity of the compound was tested against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145687(CHEMBL80680 | [(S)-[(S)-2-((R)-2-Benzyloxycarbonyl...)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibitory activity of the compound was tested against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibitory activity of the compound was tested against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  7.90E+4nMAssay Description:Inhibitory activity of the compound was tested against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)