Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50014664
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145742BDBM50145742((R)-1-(2,4-Dichloro-phenylamino)-4-pyridin-4-yl-1-...)
Affinity DataKi:  154nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145735BDBM50145735(1-(2-Bromo-phenyl)-1-(2,4-dichloro-phenylamino)-4-...)
Affinity DataKi:  204nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145751BDBM50145751((R)-1-(2-Chloro-4-methyl-phenylamino)-4-pyridin-4-...)
Affinity DataKi:  244nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145754BDBM50145754(1-(2,4-Dichloro-phenylamino)-1-(2-ethyl-phenyl)-4-...)
Affinity DataKi:  330nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145731BDBM50145731(1-(2,4-Dichloro-phenylamino)-1-(2,6-dimethyl-pheny...)
Affinity DataKi:  338nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145749BDBM50145749(1-(2,4-Dichloro-phenylamino)-4-pyridin-4-yl-1-o-to...)
Affinity DataKi:  370nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145732BDBM50145732(2-(2,4-Dichloro-phenylamino)-1-(3-hydroxy-4-methox...)
Affinity DataKi:  387nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145745BDBM50145745(1-(2-Fluoro-4-methyl-phenylamino)-4-pyridin-4-yl-1...)
Affinity DataKi:  439nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145758BDBM50145758(1-(4-Chloro-2-trifluoromethyl-phenylamino)-4-pyrid...)
Affinity DataKi:  469nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145733BDBM50145733(1-(2,4-Dichloro-phenylamino)-1-(4-fluoro-2-methyl-...)
Affinity DataKi:  512nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145739BDBM50145739(N-{3-[2-(2-Bromo-phenyl)-2-(2,4-dichloro-phenylami...)
Affinity DataKi:  514nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145741BDBM50145741((R)-1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenyl...)
Affinity DataKi:  546nMAssay Description:Binding affinity of compound towards human corticotropin releasing factor (h-CRF1) receptor showed a 2-fold activity in racemic mixtureMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145755BDBM50145755(1-(4-Methyl-2-trifluoromethyl-phenylamino)-4-pyrid...)
Affinity DataKi:  641nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145740BDBM50145740(1-(2-Chloro-4-methyl-phenylamino)-4-pyridin-4-yl-1...)
Affinity DataKi:  752nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145729BDBM50145729(1-(2-Chloro-4-methyl-phenylamino)-4-pyridin-4-yl-1...)
Affinity DataKi:  922nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145759BDBM50145759(1-(2,4-Dichloro-phenylamino)-4-pyridin-4-yl-1-(2-t...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145730BDBM50145730(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi:  1.04E+3nMAssay Description:Binding affinity of compound towards human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145737BDBM50145737(2-(2-Bromo-phenyl)-2-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145764BDBM50145764(3-[2-(2-Bromo-phenyl)-2-(2-chloro-4-methyl-phenyla...)
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145761BDBM50145761((S)-1-(2,4-Dichloro-phenylamino)-4-pyridin-4-yl-1-...)
Affinity DataKi:  3.18E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145728BDBM50145728(1-(2-Chloro-4-methyl-phenylamino)-1-(2-isopropyl-p...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145752BDBM50145752(1-(2-Chloro-4-methyl-phenylamino)-1-(2-chloro-phen...)
Affinity DataKi:  3.35E+3nMAssay Description:Binding affinity of compound towards human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145753BDBM50145753(1-(2-Chloro-4-methyl-phenylamino)-1-(3-chloro-phen...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145763BDBM50145763(1-(2-Bromo-phenyl)-1-(2-chloro-phenylamino)-4-pyri...)
Affinity DataKi:  7.33E+3nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145744BDBM50145744(1-(2-Chloro-4-methyl-phenylamino)-1-(3-methoxy-phe...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145743BDBM50145743(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145738BDBM50145738(1-(2-Chloro-4-methyl-phenylamino)-1-(2-methoxy-phe...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145736BDBM50145736(1-(2-Chloro-4-methyl-phenylamino)-1-(2-fluoro-phen...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of compound towards human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145765BDBM50145765(1-(2-Chloro-4-methyl-phenylamino)-1-phenyl-4-pyrid...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145734BDBM50145734(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145766BDBM50145766(1-(2-Chloro-4-methyl-phenylamino)-1-(4-chloro-phen...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145760BDBM50145760(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145756BDBM50145756(1-(2-Chloro-4-methyl-phenylamino)-1-(2,6-dimethoxy...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145727BDBM50145727(2-(2,4-Dichloro-phenylamino)-1-(3-hydroxy-phenyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145726BDBM50145726(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145757BDBM50145757(1-(2-Chloro-4-methyl-phenylamino)-4-pyridin-4-yl-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145725BDBM50145725(1-(2-Chloro-4-methyl-phenylamino)-1-(2,5-dimethoxy...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145724BDBM50145724(1-(2-Bromo-phenyl)-1-[(2-chloro-phenyl)-methyl-ami...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145762BDBM50145762(1-(2-Chloro-4-methyl-phenylamino)-1-(2,4-dimethoxy...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145750BDBM50145750(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145747BDBM50145747(2-(2,4-Dichloro-phenylamino)-1-(3,4-dimethoxy-phen...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145746BDBM50145746(1-(2-Chloro-4-methyl-phenylamino)-4-pyridin-4-yl-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharma Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145748BDBM50145748(1-(2-Bromo-phenyl)-1-(2-chloro-4-methyl-phenylamin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human corticotropin releasing factor (h-CRF1) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed