Compile Data Set for Download or QSAR
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Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50014672
TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145950((Z)-4-{3-[[3-(3-Carboxy-3-hydroxy-acryloyl)-phenyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145954((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145948((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145958((Z)-4-(3-{2-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  300nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145952((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-1-(4-{4-[3-(2-f...)
Affinity DataIC50:  300nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50095515(4-[3-(2-Fluoro-benzyl)-phenyl]-2,4-dioxo-butyric a...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145957((Z)-4-(3-{3-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM23399(4-{1-[(4-fluorophenyl)methyl]-1H-pyrrol-2-yl}-2,4-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145953((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  700nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145956((Z)-4-(3-{4-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  1.70E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145950((Z)-4-{3-[[3-(3-Carboxy-3-hydroxy-acryloyl)-phenyl...)
Affinity DataIC50:  1.80E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145958((Z)-4-(3-{2-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  1.80E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145956((Z)-4-(3-{4-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145952((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-1-(4-{4-[3-(2-f...)
Affinity DataIC50:  2.50E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50095515(4-[3-(2-Fluoro-benzyl)-phenyl]-2,4-dioxo-butyric a...)
Affinity DataIC50:  2.50E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145955((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145953((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  4.80E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145954((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  5.30E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145948((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  5.80E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145957((Z)-4-(3-{3-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)
Affinity DataIC50:  7.30E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM23399(4-{1-[(4-fluorophenyl)methyl]-1H-pyrrol-2-yl}-2,4-...)
Affinity DataIC50:  1.45E+4nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetIntegrase(Human immunodeficiency virus type 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145955((Z)-4-[3-(2-Fluoro-benzyl)-phenyl]-2-hydroxy-4-oxo...)
Affinity DataIC50:  3.20E+4nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed