TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Homo sapiens (Human))
Tokyo University Of Science
Curated by ChEMBL
Tokyo University Of Science
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human gamma-secretase activityMore data for this Ligand-Target Pair