Compile Data Set for Download or QSAR
Report error Found 124 Enz. Inhib. hit(s) with all data for entry = 50014918
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117232BDBM50117232(5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine |...)
Affinity DataIC50: 0.25nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117238BDBM50117238(5-Butyl-8-(4-chloro-phenyl)-3H-[1,2,4]triazolo[5,1...)
Affinity DataIC50: 0.410nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117215BDBM50117215(5-Butyl-8-(4-trifluoromethyl-phenyl)-3H-[1,2,4]tri...)
Affinity DataIC50: 0.610nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149106BDBM50149106(8-Biphenyl-4-yl-5-(2-methoxy-ethyl)-3H-[1,2,4]tria...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149112BDBM50149112(5-Butyl-2-(4-fluoro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145230BDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 2.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149110BDBM50149110(5-Butyl-2-p-tolyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 4nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149105BDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 4.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149126BDBM50149126(5-Butyl-2-(4-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117219BDBM50117219(8-Biphenyl-4-yl-5-butyl-3H-[1,2,4]triazolo[5,1-i]p...)
Affinity DataIC50: 5nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149124BDBM50149124(4-[8-(4-Chloro-phenyl)-3H-[1,2,4]triazolo[5,1-i]pu...)
Affinity DataIC50: 5.40nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149118BDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 6.20nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149122BDBM50149122(2-(4-Bromo-phenyl)-5-butyl-[1,2,4]triazolo[1,5-c]q...)
Affinity DataIC50: 8.20nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149129BDBM50149129(4-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 8.70nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149132BDBM50149132(5-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 9.10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149120BDBM50149120(5-Butyl-2-(2-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149116BDBM50149116(4-(5-Butyl-[1,2,4]triazolo[1,5-c]quinazolin-2-yl)-...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145227BDBM50145227(5-Butyl-2-(4-methoxy-phenyl)-7H-pyrazolo[4,3-e][1,...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149117BDBM50149117(5-Butyl-2-(3-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149136BDBM50149136(5-Butyl-2-(4-ethoxy-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 10nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149121BDBM50149121(5-Butyl-2-(4-ethyl-phenyl)-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 12nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149127BDBM50149127(3-(8-Biphenyl-4-yl-3H-[1,2,4]triazolo[5,1-i]purin-...)
Affinity DataIC50: 15nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149128BDBM50149128(2-(4-Bromo-phenyl)-5-butyl-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50: 19nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149130BDBM50149130(2-(4-Bromo-phenyl)-5-butyl-9-chloro-[1,2,4]triazol...)
Affinity DataIC50: 22nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149111BDBM50149111(5-Butyl-2-(4-chloro-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 26nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145230BDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 27nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149118BDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 27nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149104BDBM50149104(5-Butyl-9-chloro-2-(4-chloro-phenyl)-[1,2,4]triazo...)
Affinity DataIC50: 28nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149108BDBM50149108(5-Butyl-2-(4-fluoro-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 28nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149103BDBM50149103(5-Butyl-9-chloro-2-(4-methoxy-phenyl)-[1,2,4]triaz...)
Affinity DataIC50: 33nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149133BDBM50149133(5-Butyl-8-chloro-2-(4-methoxy-phenyl)-[1,2,4]triaz...)
Affinity DataIC50: 34nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149107BDBM50149107(5-Butyl-2-p-tolyl-[1,2,4]triazolo[1,5-c]quinazolin...)
Affinity DataIC50: 34nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149113BDBM50149113(5-Butyl-2-(4-ethoxy-phenyl)-[1,2,4]triazolo[1,5-c]...)
Affinity DataIC50: 35nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149105BDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 38nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149134BDBM50149134(5-Butyl-2-(4-propyl-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 42nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149123BDBM50149123(5-Butyl-9-chloro-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 45nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149115BDBM50149115(5-Butyl-8-chloro-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 48nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117232BDBM50117232(5-Butyl-8-phenyl-3H-[1,2,4]triazolo[5,1-i]purine |...)
Affinity DataIC50: 71nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149118BDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 100nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A2B receptor expressed in HEK293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149119BDBM50149119(5-Butyl-8-methyl-2-phenyl-[1,2,4]triazolo[1,5-c]qu...)
Affinity DataIC50: 110nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149135BDBM50149135(5-Butyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazo...)
Affinity DataIC50: 120nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149105BDBM50149105(2-Phenyl-5-propyl-7H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataIC50: 120nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145228BDBM50145228(5-Butyl-2-(4-trifluoromethyl-phenyl)-7H-pyrazolo[4...)
Affinity DataIC50: 130nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149120BDBM50149120(5-Butyl-2-(2-chloro-phenyl)-7H-pyrazolo[4,3-e][1,2...)
Affinity DataIC50: 130nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149137BDBM50149137(2-Biphenyl-4-yl-5-butyl-[1,2,4]triazolo[1,5-c]quin...)
Affinity DataIC50: 140nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149131BDBM50149131(5-Butyl-2-(4-tert-butyl-phenyl)-7H-pyrazolo[4,3-e]...)
Affinity DataIC50: 150nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145231BDBM50145231(5-Butyl-2-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-c...)
Affinity DataIC50: 160nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145230BDBM50145230(5-Butyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 190nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50145226BDBM50145226(5-Butyl-2-phenyl-[1,2,4]triazolo[1,5-c]quinazoline...)
Affinity DataIC50: 260nMAssay Description:Displacement of specific [125I]AB-MECA binding at human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50149118BDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: 310nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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