Compile Data Set for Download or QSAR
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Found 11 Enz. Inhib. hit(s) with all data for entry = 50036037
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  200nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  600nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50004771(1-(2-Amino-3-phenyl-propionyl)-pyrrolidine-2-carbo...)
Affinity DataKi:  1.30E+3nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368382(CHEMBL1202122)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368381(CHEMBL1202107)
Affinity DataKi:  2.28E+3nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368380(CHEMBL1202123)
Affinity DataKi:  1.16E+4nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368383(CHEMBL1202121)
Affinity DataKi:  1.35E+4nMAssay Description:In vitro inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  1.49E+5nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  1.57E+5nMAssay Description:In vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  1.99E+5nMAssay Description:In vitro inhibitory activity against KallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Thrombosis Research Institute

Curated by ChEMBL
LigandPNGBDBM50368379(CHEMBL1202120)
Affinity DataKi:  4.94E+5nMAssay Description:In vitro inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed