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Found 15 Enz. Inhib. hit(s) with all data for entry = 50015151
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152197(2-[3-(5-Aminomethyl-2,4-dimethyl-benzylamino)-5-ch...)
Affinity DataKi:  93nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152198(2-[3-(4-Amino-cyclohexylamino)-5-chloro-6-methyl-2...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM16127(2,2 -methanediylbis(1H-benzimidazole-6-carboximida...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152202(2-[3-(4-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  245nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152200(CHEMBL183528 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152205(2-[3-(3-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  390nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152206(CHEMBL187587 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  426nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152196(CHEMBL184815 | N-(3-Aminomethyl-phenyl)-2-{5-chlor...)
Affinity DataKi:  518nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152193(CHEMBL187649 | N-(3-Aminomethyl-phenyl)-2-{3-[(6-a...)
Affinity DataKi:  580nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152203(2-[3-(4-Aminomethyl-benzylamino)-5-chloro-6-methyl...)
Affinity DataKi:  615nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152194(2-[3-(2-Amino-benzylamino)-5-chloro-6-methyl-2-oxo...)
Affinity DataKi:  875nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152204(CHEMBL360210 | N-(3-Aminomethyl-phenyl)-2-[5-chlor...)
Affinity DataKi:  970nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152195(CHEMBL187168 | N-(3-Aminomethyl-phenyl)-2-[3-(4-be...)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152199(CHEMBL183942 | N-(3-Aminomethyl-phenyl)-2-(5-chlor...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50152201(CHEMBL187651 | N-(3-Aminomethyl-phenyl)-2-[5-chlor...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed