Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50015255
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153502(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153508(Benzo[b]thiophen-3-yl-[(4aR,5S)-1-(4-fluoro-phenyl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153504(CHEMBL366093 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153507(CHEMBL186948 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153519(CHEMBL186954 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153515(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataIC50:  5nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153503(3-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153511(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153514(4-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153506((4-Chloro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataIC50:  7nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153509(CHEMBL181601 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153513(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153501((4-Fluoro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataIC50:  9.20nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153510(CHEMBL360248 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  14nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153517(CHEMBL182827 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataIC50:  15.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153518(5-(Benzo[b]thiophen-3-yl-hydroxy-methyl)-4a-methyl...)
Affinity DataIC50:  165nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153505(5-[Hydroxy-(3,4,5-trimethoxy-phenyl)-methyl]-4a-me...)
Affinity DataIC50: >2.00E+3nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153516(5-(Hydroxy-phenyl-methyl)-4a-methyl-4,4a,5,6,7,8-h...)
Affinity DataIC50:  2.10E+3nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153501((4-Fluoro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataEC50:  8nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153504(CHEMBL366093 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  4nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153508(Benzo[b]thiophen-3-yl-[(4aR,5S)-1-(4-fluoro-phenyl...)
Affinity DataEC50:  1.80nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153506((4-Chloro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataEC50:  3nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153507(CHEMBL186948 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  3nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153509(CHEMBL181601 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  4nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153507(CHEMBL186948 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  22nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153501((4-Fluoro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataEC50:  3nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153506((4-Chloro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataEC50:  4nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153511(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  17nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.200nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153510(CHEMBL360248 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  24nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153515(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  6nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153503(3-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataEC50:  3nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153514(4-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153514(4-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataEC50:  16nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153513(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  7nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153502(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  8nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153511(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  9nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153514(4-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataEC50:  12nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153508(Benzo[b]thiophen-3-yl-[(4aR,5S)-1-(4-fluoro-phenyl...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153506((4-Chloro-phenyl)-[(4aR,5S)-1-(4-fluoro-phenyl)-4a...)
Affinity DataEC50:  9nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153513(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  11nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153515(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  4nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153513(1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6...)
Affinity DataEC50:  3nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.300nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.200nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153503(3-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,...)
Affinity DataEC50:  3nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153510(CHEMBL360248 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  31nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153510(CHEMBL360248 | [(4aR,5S)-1-(4-Fluoro-phenyl)-4a-me...)
Affinity DataEC50:  31nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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