Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50024447
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269746(CHEMBL524883 | methyl (1S,5S,11S,17S,20S,23S,29S,3...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269738(BI-32169 | CHEMBL526383)
Affinity DataIC50:  440nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269745(CHEMBL463175 | Cephalochromin | cid_160115)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed