Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50015288
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50236430((R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-...)
Affinity DataIC50:  180nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153950(CHEMBL365681 | N-{[(R)-1-(4-Chloro-benzyl)-pyrroli...)
Affinity DataIC50:  370nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50:  570nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50:  570nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153938(CHEMBL181432 | N-{[1-(4-Chloro-benzyl)-piperidin-3...)
Affinity DataIC50:  660nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153942(CHEMBL435499 | N-({[1-(4-Chloro-benzyl)-piperidin-...)
Affinity DataIC50:  700nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153917(3-{1-Hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]...)
Affinity DataIC50:  710nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409951(CHEMBL2096789)
Affinity DataIC50:  1.20E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153945(CHEMBL365854 | N-({[1-(4-Chloro-benzyl)-pyrrolidin...)
Affinity DataIC50:  2.30E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153940(CHEMBL187469 | N-({[1-(4-Chloro-benzyl)-piperidin-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153955(CHEMBL363908 | N-{[1-(4-Chloro-benzyl)-pyrrolidin-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153926(4-Methyl-thiophene-2-carboxylic acid N''-{2-[4-(4-...)
Affinity DataIC50:  7.40E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153954(4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(4-...)
Affinity DataIC50:  7.80E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153960(CHEMBL183681 | N-({[1-(4-Chloro-benzyl)-piperidin-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153959(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153952(CHEMBL186878 | N-({[1-(4-Chloro-benzyl)-pyrrolidin...)
Affinity DataIC50:  1.40E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153951(CHEMBL362780 | N-{[1-(4-Chloro-benzyl)-piperidin-3...)
Affinity DataIC50:  1.70E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153948(4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(3,...)
Affinity DataIC50:  1.70E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153943(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50:  1.90E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153939(CHEMBL187237 | N-{2-[1-(4-Chloro-benzyl)-pyrrolidi...)
Affinity DataIC50:  2.20E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153941(4-Methyl-thiophene-2-carboxylic acid N''-(2-{2-[(3...)
Affinity DataIC50:  2.60E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153946(4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(3,...)
Affinity DataIC50:  3.30E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153958(CHEMBL185283 | N-(2-{[1-(4-Chloro-benzyl)-pyrrolid...)
Affinity DataIC50:  4.00E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153949(4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(4-...)
Affinity DataIC50:  4.10E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153944(CHEMBL188170 | N-{[1-(4-Chloro-benzyl)-pyrrolidin-...)
Affinity DataIC50:  4.20E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153957(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50:  5.00E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153956(CHEMBL185190 | N-(2-{[1-(4-Chloro-benzyl)-piperidi...)
Affinity DataIC50:  6.40E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153947(CHEMBL184474 | N-({[1-(4-Chloro-benzyl)-pyrrolidin...)
Affinity DataIC50:  6.60E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153953(CHEMBL364405 | N-{2-[1-(4-Chloro-benzyl)-piperidin...)
Affinity DataIC50:  7.40E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153961(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50:  8.70E+4nMAssay Description:Concentration required to inhibit [125I]-MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153942(CHEMBL435499 | N-({[1-(4-Chloro-benzyl)-piperidin-...)
Affinity DataEC50:  40nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153938(CHEMBL181432 | N-{[1-(4-Chloro-benzyl)-piperidin-3...)
Affinity DataEC50:  610nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50236430((R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-...)
Affinity DataEC50:  20nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409951(CHEMBL2096789)
Affinity DataEC50:  360nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed