Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50015299
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154170BDBM50154170([1-(6-Chloro-1H-indazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154167BDBM50154167([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154165BDBM50154165([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154148BDBM50154148([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154174BDBM50154174([1-(1-Methyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 3.40nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154149BDBM50154149([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154149BDBM50154149([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154168BDBM50154168([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 10nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154173BDBM50154173([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154156BDBM50154156([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 18nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154155BDBM50154155([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154171BDBM50154171([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 22nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154147BDBM50154147([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154159BDBM50154159([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 36nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154163BDBM50154163([1-(2-Cyclobutyl-2H-pyrazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50: 45nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154160BDBM50154160([1-(2-Cyclopropylmethyl-2H-pyrazol-3-ylaminooxalyl...)
Affinity DataIC50: 51nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154175BDBM50154175([1-(2-Ethyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-ca...)
Affinity DataIC50: 52nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154172BDBM50154172([1-(2-Isopropyl-2H-pyrazol-3-ylaminooxalyl)-pentyl...)
Affinity DataIC50: 54nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154146BDBM50154146([1-(2-Cyclohexyl-2H-pyrazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50: 58nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154169BDBM50154169([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 62nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154176BDBM50154176([1-(2-Phenyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 63nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154162BDBM50154162([1-(2-Benzyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 65nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154164BDBM50154164([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154157BDBM50154157([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154151BDBM50154151([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154150BDBM50154150({1-[2-(3,3-Dimethyl-butyl)-2H-pyrazol-3-ylaminooxa...)
Affinity DataIC50: 71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154153BDBM50154153([1-(2-Isobutyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]...)
Affinity DataIC50: 76nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154152BDBM50154152([1-(2-Cyclopentyl-2H-pyrazol-3-ylaminooxalyl)-pent...)
Affinity DataIC50: 83nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154166BDBM50154166([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 120nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154158BDBM50154158([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 135nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154145BDBM50154145([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 140nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154154BDBM50154154([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 350nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154161BDBM50154161([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed