Compile Data Set for Download or QSAR
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Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50015328
TargetCytoplasmic protein NCK1(Human)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataEC50:  1.50E+5nMAssay Description:Displacement of PRP-1 peptide from human Nck kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154591(6-Bromo-quinolin-2-ylamine | CHEMBL189197)
Affinity DataEC50:  5.80E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataKd:  1.25E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataKd:  6.10E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154584(6-Fluoro-quinolin-2-ylamine | CHEMBL185917)
Affinity DataEC50:  1.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154585(CHEMBL187951 | Quinazolin-2-ylamine)
Affinity DataKd:  8.00E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154586(6-(5,5-Dimethyl-[1,3]dioxan-2-yl)-quinolin-2-ylami...)
Affinity DataKd:  2.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase HCK(Human)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataEC50: >1.00E+6nMAssay Description:Displacement of PRP-2 peptide from human Hck kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataEC50:  7.50E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCytoplasmic protein NCK1(Human)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataEC50: >5.00E+5nMAssay Description:Displacement of PRP-1 peptide from human Nck kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCytoplasmic protein NCK1(Human)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataEC50:  9.00E+4nMAssay Description:Displacement of PRP-1 peptide from human Nck kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataEC50:  1.60E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14320(1-amino-isoquinoline | CHEMBL62083 | Fragment 17 |...)
Affinity DataKd:  6.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCytoplasmic protein NCK1(Human)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataEC50:  3.00E+5nMAssay Description:Displacement of PRP-1 peptide from human Nck kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50013712(2-aminopyridin | 2-aminopyridine | CHEMBL21619 | P...)
Affinity DataKd: >4.00E+6nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataKd:  4.00E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50084506(CHEMBL319543 | Methyl-quinolin-2-yl-amine)
Affinity DataKd:  3.80E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154588(5,6,7,8-Tetrahydro-quinolin-2-ylamine | CHEMBL1888...)
Affinity DataEC50:  2.15E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154590(6-Methoxy-quinolin-2-ylamine | CHEMBL188730)
Affinity DataEC50:  6.30E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154589(6-Chloro-quinolin-2-ylamine | CHEMBL189514)
Affinity DataEC50:  7.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataEC50:  3.40E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataKd:  5.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataEC50:  2.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed