Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 1628
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12777BDBM12777(N-[4-(1H-1,3-benzodiazol-1-yl)-2-fluorophenyl]-2-(...)
Affinity DataKi:  2.5nM ΔG°:  -48.6kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12787BDBM12787(3-(4-aminophenyl)-N-[4-(1H-1,3-benzodiazol-1-yl)ph...)
Affinity DataKi:  4nM ΔG°:  -47.5kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12828BDBM12828(2,2,2-trifluoroacetic acid; methyl (1R,2S)-2-[2-(5...)
Affinity DataKi:  19nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12806BDBM12806(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  22nM ΔG°:  -43.3kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12802BDBM12802(2,2,2-trifluoroacetic acid; 3-(4-aminophenyl)-N-[4...)
Affinity DataKi:  47nM ΔG°:  -41.4kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12777BDBM12777(N-[4-(1H-1,3-benzodiazol-1-yl)-2-fluorophenyl]-2-(...)
Affinity DataKi:  63nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12825BDBM12825(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  65nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12805BDBM12805(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  71nM ΔG°:  -40.4kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12802BDBM12802(2,2,2-trifluoroacetic acid; 3-(4-aminophenyl)-N-[4...)
Affinity DataKi:  74nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12787BDBM12787(3-(4-aminophenyl)-N-[4-(1H-1,3-benzodiazol-1-yl)ph...)
Affinity DataKi:  75nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12818BDBM12818(2,2,2-trifluoroacetic acid; methyl (1R,2S)-2-[2-(5...)
Affinity DataKi:  90nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12800BDBM12800(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  98nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12823BDBM12823(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(5-...)
Affinity DataKi:  120nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12800BDBM12800(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  120nM ΔG°:  -39.1kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12824BDBM12824((1R,2S)-2-[2-(5-carbamimidoyl-1-benzothiophen-3-yl...)
Affinity DataKi:  130nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12815BDBM12815(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  130nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12823BDBM12823(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(5-...)
Affinity DataKi:  180nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12827BDBM12827((1R,2S)-2-[2-(5-carbamimidoyl-1-benzothiophen-3-yl...)
Affinity DataKi:  200nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12805BDBM12805(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  220nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12804BDBM12804(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  230nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12831BDBM12831(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(7-...)
Affinity DataKi:  240nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12810BDBM12810(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  250nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12829BDBM12829(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(5-...)
Affinity DataKi:  270nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12819BDBM12819(2,2,2-trifluoroacetic acid; methyl (1S,2R)-2-[(2R)...)
Affinity DataKi:  270nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12819BDBM12819(2,2,2-trifluoroacetic acid; methyl (1S,2R)-2-[(2R)...)
Affinity DataKi:  280nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12807BDBM12807(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  280nM ΔG°:  -37.0kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12825BDBM12825(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  280nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12817BDBM12817(2,2,2-trifluoroacetic acid; methyl (1S,2R)-2-[2-(5...)
Affinity DataKi:  300nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12817BDBM12817(2,2,2-trifluoroacetic acid; methyl (1S,2R)-2-[2-(5...)
Affinity DataKi:  310nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12828BDBM12828(2,2,2-trifluoroacetic acid; methyl (1R,2S)-2-[2-(5...)
Affinity DataKi:  340nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12808BDBM12808(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  390nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12815BDBM12815(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  410nM ΔG°:  -36.1kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12824BDBM12824((1R,2S)-2-[2-(5-carbamimidoyl-1-benzothiophen-3-yl...)
Affinity DataKi:  430nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12810BDBM12810(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  450nM ΔG°:  -35.9kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12821BDBM12821(R-(-) | (2R)-N-(1,3-benzothiazol-6-yl)-2-(5-carbam...)
Affinity DataKi:  480nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12818BDBM12818(2,2,2-trifluoroacetic acid; methyl (1R,2S)-2-[2-(5...)
Affinity DataKi:  500nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12831BDBM12831(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(7-...)
Affinity DataKi:  530nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12814BDBM12814(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  580nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12804BDBM12804(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  740nM ΔG°:  -34.6kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12811BDBM12811(2,2,2-trifluoroacetic acid; N-(1,3-benzothiazol-6-...)
Affinity DataKi:  780nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12811BDBM12811(2,2,2-trifluoroacetic acid; N-(1,3-benzothiazol-6-...)
Affinity DataKi:  780nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12809BDBM12809(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  930nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12813BDBM12813(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  960nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12829BDBM12829(2,2,2-trifluoroacetic acid; ethyl (1R,2S)-2-[2-(5-...)
Affinity DataKi:  1.19E+3nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12807BDBM12807(2,2,2-trifluoroacetic acid; N-[4-(1H-1,3-benzodiaz...)
Affinity DataKi:  1.25E+3nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12812BDBM12812(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  1.73E+3nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12808BDBM12808(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  2.02E+3nM ΔG°:  -32.2kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12821BDBM12821(R-(-) | (2R)-N-(1,3-benzothiazol-6-yl)-2-(5-carbam...)
Affinity DataKi:  2.70E+3nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12814BDBM12814(2,2,2-trifluoroacetic acid; 2-(5-carbamimidoyl-1-b...)
Affinity DataKi:  3.24E+3nM ΔG°:  -31.0kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandChemical structure of BindingDB Monomer ID 12827BDBM12827((1R,2S)-2-[2-(5-carbamimidoyl-1-benzothiophen-3-yl...)
Affinity DataKi:  3.50E+3nMAssay Description:Ki values were obtained from human purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were deter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2007
Entry Details Article
PubMed
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