Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50015626
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  2nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158497(2-benzo[b]thiophen-3-yl-N-[1-(3,4-dichlorobenzyl)p...)
Affinity DataKi:  360nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158501(CHEMBL224686 | N-[1-(3,4-dichlorobenzyl)pyrrolidin...)
Affinity DataKi:  510nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158498(2-benzo[1,3]dioxol-5-yl-N-[1-(3,4-dichlorobenzyl)p...)
Affinity DataKi:  630nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158502(CHEMBL224519 | N-[1-(3,4-dichlorobenzyl)pyrrolidin...)
Affinity DataKi:  980nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158495(CHEMBL224943 | [5-(4-chlorophenyl)furan-2-ylmethyl...)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158496((R)-N-(1-phenethylpyrrolidin-2-ylmethyl)-4-phenylb...)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158499(CHEMBL225073 | [5-(4-chlorophenyl)-furan-2-ylmethy...)
Affinity DataKi:  5.00E+3nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50411328(CHEMBL2096864)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158494((R)-2-benzo[b]thiophen-3-yl-N-[1-(3,4-dichlorobenz...)
Affinity DataKi:  9.80E+3nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158504(CHEMBL387725 | N-(1-benzylpyrrolidin-3-yl)-2-pheny...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158503(CHEMBL224518 | N-(1-phenethylpyrrolidin-3-yl)-2-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50411329(CHEMBL2096865)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50158500(CHEMBL224219 | N-(1-(3,4-dichlorobenzyl)pyrrolidin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed