Compile Data Set for Download or QSAR
Report error Found 126 Enz. Inhib. hit(s) with all data for entry = 50015642
LigandChemical structure of BindingDB Monomer ID 20464BDBM20464((2E)-3-[2-(piperidin-1-yl)-6-(trifluoromethyl)pyri...)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 20464BDBM20464((2E)-3-[2-(piperidin-1-yl)-6-(trifluoromethyl)pyri...)
Affinity DataIC50: 1nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158665BDBM50158665(3-(4-tert-butylphenyl)-N-(quinolin-7-yl)acrylamide...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158658BDBM50158658((E)-3-(2-Morpholin-4-yl-6-trifluoromethyl-pyridin-...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158658BDBM50158658((E)-3-(2-Morpholin-4-yl-6-trifluoromethyl-pyridin-...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158665BDBM50158665(3-(4-tert-butylphenyl)-N-(quinolin-7-yl)acrylamide...)
Affinity DataIC50: 2nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158681BDBM50158681((E)-3-(4-tert-Butyl-phenyl)-N-(2-oxo-1,2,3,4-tetra...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158679BDBM50158679((E)-3-(4-tert-Butyl-phenyl)-N-(3-oxo-3,4-dihydro-2...)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158678BDBM50158678(3-(4-tert-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4]...)
Affinity DataIC50: 14nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158628BDBM50158628(ethyl 5-tert-butyl-2-(3-(2,3-dihydrobenzo[b][1,4]d...)
Affinity DataIC50: 15nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158647BDBM50158647((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2-mor...)
Affinity DataIC50: 15nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158683BDBM50158683(3-(4-tert-butylphenyl)-N-(3,4-dihydro-2H-benzo[b][...)
Affinity DataIC50: 16nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158633BDBM50158633((E)-3-(4-tert-Butyl-phenyl)-5-methyl-hex-2-enoic a...)
Affinity DataIC50: 16nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158634BDBM50158634(3-(4-tert-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4]...)
Affinity DataIC50: 20nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158671BDBM50158671((E)-3-(4-tert-Butyl-phenyl)-N-(3-methoxy-phenyl)-a...)
Affinity DataIC50: 21nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158655BDBM50158655((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 25nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158628BDBM50158628(ethyl 5-tert-butyl-2-(3-(2,3-dihydrobenzo[b][1,4]d...)
Affinity DataIC50: 26nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158649BDBM50158649((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(6''-t...)
Affinity DataIC50: 27nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158640BDBM50158640((E)-3-(4-tert-Butyl-phenyl)-N-(3-hydroxy-4-methoxy...)
Affinity DataIC50: 30nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158646BDBM50158646((E)-4-(4-tert-Butyl-phenyl)-5-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 36nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158630BDBM50158630((E)-3-(4-tert-Butyl-phenyl)-N-(1,2,3,4-tetrahydro-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158664BDBM50158664((E)-3-(4-tert-Butyl-phenyl)-but-2-enoic acid (2,3-...)
Affinity DataIC50: 39nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158647BDBM50158647((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2-mor...)
Affinity DataIC50: 40nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158632BDBM50158632((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 44nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158666BDBM50158666((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-tri...)
Affinity DataIC50: 46nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158649BDBM50158649((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(6''-t...)
Affinity DataIC50: 54nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158668BDBM50158668(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-(4-isopr...)
Affinity DataIC50: 55nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158683BDBM50158683(3-(4-tert-butylphenyl)-N-(3,4-dihydro-2H-benzo[b][...)
Affinity DataIC50: 57nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158667BDBM50158667(3-(2-bromo-4-tert-butylphenyl)-N-(2,3-dihydrobenzo...)
Affinity DataIC50: 60nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158643BDBM50158643(3-(4-tert-butylphenyl)-N-(5,6,7,8-tetrahydronaphth...)
Affinity DataIC50: 61nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158681BDBM50158681((E)-3-(4-tert-Butyl-phenyl)-N-(2-oxo-1,2,3,4-tetra...)
Affinity DataIC50: 71nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158650BDBM50158650((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 78nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158668BDBM50158668(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-(4-isopr...)
Affinity DataIC50: 82nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158633BDBM50158633((E)-3-(4-tert-Butyl-phenyl)-5-methyl-hex-2-enoic a...)
Affinity DataIC50: 94nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158662BDBM50158662((E)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158666BDBM50158666((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-tri...)
Affinity DataIC50: 100nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158685BDBM50158685((E)-3-(6-tert-Butyl-pyridin-3-yl)-N-(2,3-dihydro-b...)
Affinity DataIC50: 100nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158682BDBM50158682(3-(4-tert-butylphenyl)-N-(3,4-dihydro-2H-benzo[b][...)
Affinity DataIC50: 110nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158636BDBM50158636((E)-3-(4-Bromo-phenyl)-N-(2,3-dihydro-benzo[1,4]di...)
Affinity DataIC50: 110nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158678BDBM50158678(3-(4-tert-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4]...)
Affinity DataIC50: 110nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158634BDBM50158634(3-(4-tert-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4]...)
Affinity DataIC50: 120nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158645BDBM50158645(3-(4-tert-butylphenyl)-N-(4-methoxyphenyl)acrylami...)
Affinity DataIC50: 140nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158644BDBM50158644(3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1,4]d...)
Affinity DataIC50: 150nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158630BDBM50158630((E)-3-(4-tert-Butyl-phenyl)-N-(1,2,3,4-tetrahydro-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158680BDBM50158680((E)-3-(4-tert-Butyl-phenyl)-N-(3,4-dimethoxy-pheny...)
Affinity DataIC50: 170nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158629BDBM50158629((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-eth...)
Affinity DataIC50: 170nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158655BDBM50158655((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50: 180nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158676BDBM50158676((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-nit...)
Affinity DataIC50: 190nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158670BDBM50158670((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-p-toly...)
Affinity DataIC50: 210nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50158674BDBM50158674(2-[1-(4-tert-Butyl-phenyl)-meth-(E)-ylidene]-N-(2,...)
Affinity DataIC50: 210nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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