Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50015644
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698(CHEMBL266078 | [N40,Pro1,Tyr4]BB)
Affinity DataIC50:  0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699(CHEMBL414307 | [(N4-Bzdig)0]BB(7-14))
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697(CHEMBL268222 | [N40,Pro1,Tyr4,Nle 14]BB)
Affinity DataIC50:  0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698(CHEMBL266078 | [N40,Pro1,Tyr4]BB)
Affinity DataIC50:  0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700(CHEMBL266079 | [(N4-Bzdig)0,Nle14]BB(7-14))
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699(CHEMBL414307 | [(N4-Bzdig)0]BB(7-14))
Affinity DataIC50:  0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158702(CHEMBL413893 | Universal ligand)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158701(CHEMBL407101 | [Tyr4]Bombesin)
Affinity DataIC50:  0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699(CHEMBL414307 | [(N4-Bzdig)0]BB(7-14))
Affinity DataIC50:  0.900nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158702(CHEMBL413893 | Universal ligand)
Affinity DataIC50:  0.960nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158702(CHEMBL413893 | Universal ligand)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700(CHEMBL266079 | [(N4-Bzdig)0,Nle14]BB(7-14))
Affinity DataIC50:  1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698(CHEMBL266078 | [N40,Pro1,Tyr4]BB)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697(CHEMBL268222 | [N40,Pro1,Tyr4,Nle 14]BB)
Affinity DataIC50:  1.94nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700(CHEMBL266079 | [(N4-Bzdig)0,Nle14]BB(7-14))
Affinity DataIC50:  2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697(CHEMBL268222 | [N40,Pro1,Tyr4,Nle 14]BB)
Affinity DataIC50:  11.2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699(CHEMBL414307 | [(N4-Bzdig)0]BB(7-14))
Affinity DataIC50:  37nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698(CHEMBL266078 | [N40,Pro1,Tyr4]BB)
Affinity DataIC50: >100nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697(CHEMBL268222 | [N40,Pro1,Tyr4,Nle 14]BB)
Affinity DataIC50: >100nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700(CHEMBL266079 | [(N4-Bzdig)0,Nle14]BB(7-14))
Affinity DataIC50: >100nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed