Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50015730
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160450BDBM50160450(1-{(S)-1-[2-(3-Chloro-phenyl)-ethyl]-piperidin-3-y...)
Affinity DataIC50: 0.600nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160449BDBM50160449(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 0.630nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160459BDBM50160459(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 1.20nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160462BDBM50160462(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 1.30nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160453BDBM50160453(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 1.60nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160482BDBM50160482(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 1.60nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160468BDBM50160468(1-{(S)-1-[2-(2,4-Difluoro-phenyl)-ethyl]-piperidin...)
Affinity DataIC50: 1.80nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160470BDBM50160470(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 1.90nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160481BDBM50160481(1-{(3S,4S)-4-Ethyl-1-[2-(4-fluoro-phenyl)-ethyl]-p...)
Affinity DataIC50: 2.20nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160476BDBM50160476(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 2.20nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160473BDBM50160473(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 3nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160455BDBM50160455(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 3nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160472BDBM50160472(1-{(S)-1-[2-(3,4-Difluoro-phenyl)-ethyl]-piperidin...)
Affinity DataIC50: 3.20nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160457BDBM50160457(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 3.40nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160457BDBM50160457(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 3.40nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160464BDBM50160464(1-{(S)-1-[2-(4-Chloro-phenyl)-ethyl]-piperidin-3-y...)
Affinity DataIC50: 3.60nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160447BDBM50160447(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 3.70nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160463BDBM50160463(1-{(S)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-y...)
Affinity DataIC50: 5nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160469BDBM50160469(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 5.5nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160458BDBM50160458(1-{(S)-1-[2-(2,4-Dichloro-phenyl)-ethyl]-piperidin...)
Affinity DataIC50: 5.5nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160456BDBM50160456(1-{(S)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-y...)
Affinity DataIC50: 6nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160466BDBM50160466(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 7.90nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160454BDBM50160454(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 9.70nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160474BDBM50160474(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 12nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160452BDBM50160452(1-{(R)-1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-3-y...)
Affinity DataIC50: 13nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160478BDBM50160478(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 14nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160479BDBM50160479(1-{(R)-1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-3-...)
Affinity DataIC50: 15nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160451BDBM50160451(1-{(S)-1-[4-(4-Fluoro-phenyl)-butyl]-piperidin-3-y...)
Affinity DataIC50: 29nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160460BDBM50160460(1-{(S)-1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-3-...)
Affinity DataIC50: 36nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160448BDBM50160448(1-[1-(4-Fluoro-benzyl)-piperidin-4-ylmethyl]-3-[3-...)
Affinity DataIC50: 54nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160471BDBM50160471(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 82nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160475BDBM50160475(1-[3-Ethyl-5-(1-methyl-1H-tetrazol-5-yl)-phenyl]-3...)
Affinity DataIC50: 120nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160467BDBM50160467(1-{1-[3-(4-Fluoro-phenyl)-propyl]-piperidin-4-ylme...)
Affinity DataIC50: 230nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160465BDBM50160465(1-{1-[2-(4-Fluoro-phenyl)-ethyl]-piperidin-4-ylmet...)
Affinity DataIC50: 350nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160461BDBM50160461(1-{(S)-1-[2-(4-Dimethylamino-phenyl)-ethyl]-piperi...)
Affinity DataIC50: 380nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
Dbristol-Myers Squibb

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160477BDBM50160477(1-[(S)-1-(4-Fluoro-benzyl)-piperidin-3-ylmethyl]-3...)
Affinity DataIC50: 3.50E+3nMAssay Description:Evaluated for inhibition of human C-C chemokine receptor type 3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed