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Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50015732
TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160523(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160523(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  4.20nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160511(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160515(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160511(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160515(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50410086(CHEMBL2096778)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160513(1-Benzyl-2-{2-[3-(2-chloro-phenyl)-ureido]-ethyl}-...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160520(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  51nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160518(1-Benzyl-2-{2-[3-(2-fluoro-phenyl)-ureido]-ethyl}-...)
Affinity DataIC50:  53nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160520(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  57nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160518(1-Benzyl-2-{2-[3-(2-fluoro-phenyl)-ureido]-ethyl}-...)
Affinity DataIC50:  66nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160522(1-Benzyl-2-[2-(3-isopropyl-ureido)-ethyl]-1H-benzo...)
Affinity DataIC50:  79nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160513(1-Benzyl-2-{2-[3-(2-chloro-phenyl)-ureido]-ethyl}-...)
Affinity DataIC50:  83nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160508(1-Benzyl-2-[3-(3-tert-butyl-ureido)-propyl]-1H-ben...)
Affinity DataIC50:  83nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50410086(CHEMBL2096778)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160519(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160488(1-Benzyl-2-(2-pyridin-3-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160488(1-Benzyl-2-(2-pyridin-3-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  140nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160522(1-Benzyl-2-[2-(3-isopropyl-ureido)-ethyl]-1H-benzo...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160519(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160508(1-Benzyl-2-[3-(3-tert-butyl-ureido)-propyl]-1H-ben...)
Affinity DataIC50:  180nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160507(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160512(4-[1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoi...)
Affinity DataIC50:  230nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160514(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  310nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160507(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160509(1-Benzyl-2-[2-(3-ethyl-ureido)-ethyl]-1H-benzoimid...)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160524(1-Benzyl-2-isopropyl-1H-benzoimidazole-5-sulfonic ...)
Affinity DataIC50:  390nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160512(4-[1-Benzyl-5-(4-fluoro-benzylsulfamoyl)-1H-benzoi...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160521(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160514(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  490nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160517(CHEMBL183197 | {2-[1-Benzyl-5-(4-fluoro-benzylsulf...)
Affinity DataIC50:  540nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160524(1-Benzyl-2-isopropyl-1H-benzoimidazole-5-sulfonic ...)
Affinity DataIC50:  690nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160509(1-Benzyl-2-[2-(3-ethyl-ureido)-ethyl]-1H-benzoimid...)
Affinity DataIC50:  690nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160517(CHEMBL183197 | {2-[1-Benzyl-5-(4-fluoro-benzylsulf...)
Affinity DataIC50:  740nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160521(1-Benzyl-2-[2-(3-tert-butyl-ureido)-ethyl]-1H-benz...)
Affinity DataIC50:  750nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160506(CHEMBL427146 | N-{2-[1-Benzyl-5-(4-fluoro-benzylsu...)
Affinity DataIC50:  840nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160510(1-Benzyl-2-cyclopropyl-1H-benzoimidazole-5-sulfoni...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160510(1-Benzyl-2-cyclopropyl-1H-benzoimidazole-5-sulfoni...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160506(CHEMBL427146 | N-{2-[1-Benzyl-5-(4-fluoro-benzylsu...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160516(2-(2-Amino-ethyl)-1-benzyl-1H-benzoimidazole-5-sul...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160516(2-(2-Amino-ethyl)-1-benzyl-1H-benzoimidazole-5-sul...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160505(1-Benzyl-2-propyl-1H-benzoimidazole-5-sulfonic aci...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration of the compound towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160505(1-Benzyl-2-propyl-1H-benzoimidazole-5-sulfonic aci...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration of the compound towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed