Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50003706
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474994BDBM50474994(Bisarylmaleimide 1)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475025BDBM50475025(CHEMBL181339)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475007BDBM50475007(Bisarylmaleimide 2)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475024BDBM50475024(CHEMBL181371)
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475018BDBM50475018(CHEMBL181518)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475031BDBM50475031(CHEMBL359871)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475029BDBM50475029(CHEMBL180779)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475008BDBM50475008(CHEMBL369090)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150698BDBM50150698(3-(imidazo[1,2-a]pyridin-3-yl)-4-(2-(morpholine-4-...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475022BDBM50475022(CHEMBL361765)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150702BDBM50150702(3-Imidazo[1,2-a]pyridin-3-yl-4-[2-(piperidine-1-ca...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474994BDBM50474994(Bisarylmaleimide 1)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150701BDBM50150701(7-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475010BDBM50475010(CHEMBL369316)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475001BDBM50475001(CHEMBL368246)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475004BDBM50475004(CHEMBL369572)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475014BDBM50475014(CHEMBL361948)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150702BDBM50150702(3-Imidazo[1,2-a]pyridin-3-yl-4-[2-(piperidine-1-ca...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475006BDBM50475006(CHEMBL178851)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474996BDBM50474996(CHEMBL178646)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475000BDBM50475000(CHEMBL181296)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150698BDBM50150698(3-(imidazo[1,2-a]pyridin-3-yl)-4-(2-(morpholine-4-...)
Affinity DataIC50: 2.60nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475011BDBM50475011(CHEMBL178850)
Affinity DataIC50: 2.70nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475021BDBM50475021(CHEMBL445649)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475009BDBM50475009(CHEMBL361635)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475016BDBM50475016(CHEMBL361007)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475005BDBM50475005(CHEMBL178820)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474993BDBM50474993(CHEMBL361996)
Affinity DataIC50: 3.40nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475028BDBM50475028(CHEMBL179725)
Affinity DataIC50: 3.5nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475020BDBM50475020(CHEMBL181464)
Affinity DataIC50: 4.70nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475027BDBM50475027(CHEMBL359537)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475001BDBM50475001(CHEMBL368246)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475025BDBM50475025(CHEMBL181339)
Affinity DataIC50: 7.70nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475006BDBM50475006(CHEMBL178851)
Affinity DataIC50: 8.70nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475016BDBM50475016(CHEMBL361007)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475030BDBM50475030(CHEMBL426243)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150701BDBM50150701(7-(4-Imidazo[1,2-a]pyridin-3-yl-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475028BDBM50475028(CHEMBL179725)
Affinity DataIC50: 13nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475015BDBM50475015(CHEMBL181774)
Affinity DataIC50: 13nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474992BDBM50474992(CHEMBL369108)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474997BDBM50474997(CHEMBL361125)
Affinity DataIC50: 27nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474998BDBM50474998(CHEMBL182048)
Affinity DataIC50: 27nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475033BDBM50475033(CHEMBL362221)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475019BDBM50475019(CHEMBL362587)
Affinity DataIC50: 33nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475023BDBM50475023(CHEMBL178645)
Affinity DataIC50: 34nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475020BDBM50475020(CHEMBL181464)
Affinity DataIC50: 38nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474995BDBM50474995(CHEMBL181015)
Affinity DataIC50: 41nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50474999BDBM50474999(CHEMBL369099)
Affinity DataIC50: 45nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475004BDBM50475004(CHEMBL369572)
Affinity DataIC50: 53nMAssay Description:Inhibitory concentration to inhibit Ser396 phosphorylation of tau, a natural substrate of GSK-3 in SY5Y cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475032BDBM50475032(CHEMBL181112)
Affinity DataIC50: 60nMAssay Description:Inhibitory concentration against the Glycogen synthase kinase-3 More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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