Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 1193
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9872BDBM9872((2S)-2-[(4-aminobenzene)(2-methylpropyl)sulfonamid...)
Affinity DataKi:  2.10nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9863BDBM9863((2S)-2-[(cyclopropylmethyl)(4-methylbenzene)sulfon...)
Affinity DataKi:  3.90nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9858BDBM9858((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  5nM ΔG°:  -48.2kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9864BDBM9864((2S)-2-[(cyclopentylmethyl)(4-methylbenzene)sulfon...)
Affinity DataKi:  5.20nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9871BDBM9871((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  7.20nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9862BDBM9862((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  13.5nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9861BDBM9861((2S)-2-[(2-ethylbutyl)(4-methylbenzene)sulfonamido...)
Affinity DataKi:  15.2nM ΔG°:  -45.4kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9869BDBM9869((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  17.4nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9865BDBM9865((2S)-2-[benzene(2-methylpropyl)sulfonamido]-6-{[(9...)
Affinity DataKi:  18.7nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9860BDBM9860((2S)-2-[benzyl(4-methylbenzene)sulfonamido]-6-{[(9...)
Affinity DataKi:  19.6nM ΔG°:  -44.7kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9870BDBM9870((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  42nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9868BDBM9868((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  54.9nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9877BDBM9877((2S)-6-[1-(9H-fluoren-9-yl)acetamido]-2-[(4-methyl...)
Affinity DataKi:  89.7nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9878BDBM9878((2S)-6-(9H-fluoren-9-ylformamido)-2-[(4-methylbenz...)
Affinity DataKi:  105nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9883BDBM9883(9H-fluoren-9-ylmethyl N-[(5S)-6-hydroxy-5-[(4-meth...)
Affinity DataKi:  105nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9884BDBM9884(9H-fluoren-9-ylmethyl N-[(5S)-5-carbamoyl-5-[(4-me...)
Affinity DataKi:  107nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9885BDBM9885(9H-fluoren-9-ylmethyl N-[(5S)-5-carbamothioyl-5-[(...)
Affinity DataKi:  127nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9873BDBM9873((2S)-5-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  180nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9887BDBM9887(9H-fluoren-9-ylmethyl N-[(5S)-5-(hydroxycarbamoyl)...)
Affinity DataKi:  245nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9874BDBM9874((2S)-7-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi: >250nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9875BDBM9875((2S)-4-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi: >250nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9876BDBM9876((2S)-3-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi: >250nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9879BDBM9879((2S)-6-{[(tert-butoxy)carbonyl]amino}-2-[(4-methyl...)
Affinity DataKi: >250nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9888BDBM9888(9H-fluoren-9-ylmethyl N-[(5S)-5-(hydrazinecarbonyl...)
Affinity DataKi:  254nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9867BDBM9867((2S)-2-[(4-tert-butylbenzene)(2-methylpropyl)sulfo...)
Affinity DataKi:  257nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9886BDBM9886(9H-fluoren-9-ylmethyl N-[(5S)-5-carbamimidoyl-5-[(...)
Affinity DataKi:  280nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9889BDBM9889(9H-fluoren-9-ylmethyl N-[(5S)-5-[(4-methylbenzene)...)
Affinity DataKi: >300nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9890BDBM9890(9H-fluoren-9-ylmethyl N-[(5S)-6-amino-5-[(4-methyl...)
Affinity DataKi: >300nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9881BDBM9881(methyl (2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]a...)
Affinity DataKi: >300nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9866BDBM9866((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi: >300nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9882BDBM9882(9H-fluoren-9-ylmethyl N-[(5S)-5-[(4-methylbenzene)...)
Affinity DataKi: >300nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9859BDBM9859((2R)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  330nM ΔG°:  -37.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9857BDBM9857((2S)-2-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-6...)
Affinity DataKi:  2.00E+3nM ΔG°:  -33.1kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9856BDBM9856((2S)-6-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-2...)
Affinity DataKi:  8.00E+3nM ΔG°:  -29.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9855BDBM9855((2S)-2-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-6...)
Affinity DataKi:  1.05E+4nM ΔG°:  -28.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9853BDBM9853((2S)-2-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-5...)
Affinity DataKi:  1.42E+4nM ΔG°:  -28.1kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9852BDBM9852((2S)-2-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-6...)
Affinity DataKi:  1.74E+4nM ΔG°:  -27.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9851BDBM9851((2S)-6-{[(benzyloxy)carbonyl]amino}-2-{[(9H-fluore...)
Affinity DataKi:  2.15E+4nM ΔG°:  -27.1kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9854BDBM9854((2S)-2-{[(9H-fluoren-9-ylmethoxy)carbonyl]amino}-5...)
Affinity DataKi:  2.62E+4nM ΔG°:  -26.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9850BDBM9850((2S)-6-{[(tert-butoxy)carbonyl]amino}-2-{[(9H-fluo...)
Affinity DataKi:  2.80E+4nM ΔG°:  -26.4kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9848BDBM9848((2S)-2-{[(benzyloxy)carbonyl]amino}-6-{[(tert-buto...)
Affinity DataKi: >1.00E+5nM ΔG°: >-23.2kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9849BDBM9849((2S)-6-{[(tert-butoxy)carbonyl]amino}-2-[(4-methyl...)
Affinity DataKi: >1.00E+5nM ΔG°: >-23.2kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2006
Entry Details Article
PubMed