Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50015957
LigandPNGBDBM50162884(3-[[2-(4-Fluoro-phenyl)-ethyl]-(4-phenoxy-benzyl)-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162889(2-[4-(2-Amino-3-mercapto-propylamino)-2-naphthalen...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162883(CHEMBL425159 | [2-(4-Bromo-phenyl)-ethyl]-(1H-imid...)
Affinity DataIC50:  256nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162888(CHEMBL426604 | [2-(4-Fluoro-phenyl)-ethyl]-(1H-imi...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162882(3-(1H-Imidazol-4-yl)-3-[(4-phenoxy-benzyl)-(4-phen...)
Affinity DataIC50:  860nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162885(3-[Biphenyl-4-ylmethyl-(2-thiophen-2-yl-ethyl)-ami...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162887(3-{(4-Butoxy-benzenesulfonyl)-[2-(4-fluoro-phenyl)...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50162886(3-{Biphenyl-4-ylmethyl-[2-(4-fluoro-phenyl)-ethyl]...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50162888(CHEMBL426604 | [2-(4-Fluoro-phenyl)-ethyl]-(1H-imi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50162883(CHEMBL425159 | [2-(4-Bromo-phenyl)-ethyl]-(1H-imid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed