Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50037435
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292221BDBM50292221((S)-3-(2,4-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366689BDBM50366689(GHRELIN)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292225BDBM50292225((S)-3-(2,5-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292228BDBM50292228((S)-3-(2,3-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151162BDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50151162BDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 4nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292230BDBM50292230((S)-3-(2,6-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292223BDBM50292223((R)-3-(3-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 15nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292227BDBM50292227((R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(3-methox...)
Affinity DataIC50: 77nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292226BDBM50292226((R)-3-(4-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 83nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292229BDBM50292229((R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(4-methox...)
Affinity DataIC50: 106nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292224BDBM50292224(1-(2-Diethylamino-ethyl)-3-hydroxy-2-oxo-3-phenyl-...)
Affinity DataIC50: 116nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292222BDBM50292222((S)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(2-methox...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed