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Found 20 Enz. Inhib. hit(s) with all data for entry = 50016020
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163887(CHEMBL183565 | N-[4-(1H-Indol-5-yloxy)-3,5-bis-tri...)
Affinity DataEC50:  23nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163906(CHEMBL361162 | [4-(3-Isopropyl-1H-indol-5-yloxy)-3...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163889(CHEMBL182430 | N-[3-Chloro-4-(3-isopropyl-1H-indol...)
Affinity DataEC50:  8nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163890(CHEMBL183050 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163891(CHEMBL360774 | N-{4-[3-(4-Fluoro-phenyl)-1H-indol-...)
Affinity DataEC50:  115nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163892(CHEMBL183851 | N-[3,5-Dimethyl-4-(3-pentyl-1H-inda...)
Affinity DataEC50:  8nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163893(CHEMBL183057 | N-[3,5-Dimethyl-4-(3-methyl-1H-indo...)
Affinity DataEC50:  15nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163895((S)-2-Amino-3-[4-(4-hydroxy-3-iodo-phenoxy)-3-iodo...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163894(CHEMBL183863 | N-{4-[3-(4-Fluoro-benzyl)-1H-indol-...)
Affinity DataEC50:  11nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163896(CHEMBL183000 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163898(CHEMBL359647 | N-[3-Chloro-4-(3-isopropyl-1H-indol...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163897(3-[4-(3-Isopropyl-1H-indol-5-yloxy)-3,5-bis-triflu...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163902(CHEMBL183727 | N-[3,5-Dichloro-4-(1H-indol-5-yloxy...)
Affinity DataEC50:  15nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163899(CHEMBL183122 | N-[3,5-Dichloro-4-(3-isopropyl-1H-i...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163900((E)-3-[4-(3-Isopropyl-1H-indol-5-yloxy)-3,5-bis-tr...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163901(CHEMBL360137 | N-[3,5-Dibromo-4-(3-isopropyl-1H-in...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163904(CHEMBL180952 | N-[4-(3-Isopropyl-1H-indol-5-ylmeth...)
Affinity DataEC50:  18nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163905(CHEMBL183829 | N-[4-(1H-Indol-5-yloxy)-3,5-dimethy...)
Affinity DataEC50:  72nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163903(CHEMBL180819 | N-{4-[3-(4-Fluoro-phenoxy)-1H-indol...)
Affinity DataEC50:  495nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163888(CHEMBL183176 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  3nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed