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Found 18 Enz. Inhib. hit(s) with all data for entry = 50016042
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(CHEMBL190022 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(CHEMBL193212 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50:  420nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224(CHEMBL192921 | {Imidazo[1,2-d][1,2,4]thiadiazol-3-...)
Affinity DataIC50:  620nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164225(CHEMBL365470 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164226(CHEMBL193724 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  910nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164218(CHEMBL192770 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164221(CHEMBL189379 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164219(CHEMBL190568 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(CHEMBL190022 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(CHEMBL193212 | N-[6-(Imidazo[1,2-d][1,2,4]thiadiaz...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164217(CHEMBL192660 | N*1*-Imidazo[1,2-d][1,2,4]thiadiazo...)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224(CHEMBL192921 | {Imidazo[1,2-d][1,2,4]thiadiazol-3-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164220(CHEMBL192376 | N-Hexyl-2-nitro-benzenesulfonamide)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164215(2-Nitro-N-[6-(3-nitro-pyridin-2-ylamino)-hexyl]-be...)
Affinity DataIC50:  1.70E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed