Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 763
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5815BDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5815BDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 3nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5825BDBM5825(3-{4-[methyl({2-[(3-sulfamoylphenyl)amino]pyrimidi...)
Affinity DataIC50: 5nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5819BDBM5819(3-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 18nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5816BDBM5816(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5814BDBM5814(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5810BDBM5810(N-{3-[4-amino-5-(4-phenylphenyl)furo[2,3-d]pyrimid...)
Affinity DataIC50: 36nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5818BDBM5818({4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidi...)
Affinity DataIC50: 58nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5817BDBM5817(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 59nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5814BDBM5814(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 62nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5808BDBM5808(N-{3-[4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 65nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5821BDBM5821(phenyl N-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]...)
Affinity DataIC50: 95nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5822BDBM5822(3-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 117nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5820BDBM5820(N-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 176nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5806BDBM5806(3-[4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin...)
Affinity DataIC50: 180nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5817BDBM5817(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 186nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5810BDBM5810(N-{3-[4-amino-5-(4-phenylphenyl)furo[2,3-d]pyrimid...)
Affinity DataIC50: 190nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5823BDBM5823(N-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 269nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5818BDBM5818({4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidi...)
Affinity DataIC50: 275nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5808BDBM5808(N-{3-[4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 300nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5824BDBM5824(1-{4-[(2-{[3-(methanesulfonylmethyl)phenyl]amino}p...)
Affinity DataIC50: 324nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5809BDBM5809(5-[4-(dimethylamino)phenyl]-6-(4-methoxyphenyl)fur...)
Affinity DataIC50: 350nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5812BDBM5812(N-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 501nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5806BDBM5806(3-[4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin...)
Affinity DataIC50: 540nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5809BDBM5809(5-[4-(dimethylamino)phenyl]-6-(4-methoxyphenyl)fur...)
Affinity DataIC50: 600nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5813BDBM5813(N-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 851nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5802BDBM5802(5,6-bis(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-ami...)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5802BDBM5802(5,6-bis(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-ami...)
Affinity DataIC50: 1.12E+3nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5807BDBM5807(3-[4-amino-5-(4-methoxyphenyl)furo[2,3-d]pyrimidin...)
Affinity DataIC50: 1.48E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5805BDBM5805(6-(3,4-dichlorophenyl)-5-(4-methoxyphenyl)furo[2,3...)
Affinity DataIC50: 1.78E+3nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5803BDBM5803(5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine | ...)
Affinity DataIC50: 5.50E+3nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5804BDBM5804(6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine | ...)
Affinity DataIC50: 1.70E+4nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5811BDBM5811(N-{3-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 2.00E+4nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5803BDBM5803(5-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine | ...)
Affinity DataIC50: 2.00E+4nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 5804BDBM5804(6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-amine | ...)
Affinity DataIC50: 2.00E+4nMpH: 7.5 T: 2°CAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 5805BDBM5805(6-(3,4-dichlorophenyl)-5-(4-methoxyphenyl)furo[2,3...)
Affinity DataIC50: 2.00E+4nMAssay Description:The assay was using baculovirus-expressed recombinant protein kinase purified as the intracellular domain fused by GST tag, interacting with biotinyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2005
Entry Details Article
PubMed