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Found 11 Enz. Inhib. hit(s) with all data for entry = 50016144
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50:  400nMAssay Description:Mean inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50:  790nMAssay Description:Mean inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50:  1.32E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50:  3.16E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50:  5.29E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50:  1.05E+4nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50:  2.49E+4nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50:  1.04E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50:  1.07E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50:  1.37E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50:  1.55E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed